SCHEMBL8096036

SCHEMBL8096036

CC(C)Cc1nc(CC(C)C)n(Cc2ccc(-c3cccc(C(=O)O)c3)cc2)n1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 1/20 0.48
AGTR2 P50052 1/20 0.48
PPARG P37231 1/20 0.48
ALOX5AP P20292 2/20 0.47
PDE7A Q13946 1/20 0.43
PDE7B Q9NP56 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PTGES O14684 1/20 0.41
ALOX5 P09917 1/20 0.41
LTC4S Q16873 1/20 0.41
MGLL Q99685 1/20 0.41
DHFR P00374 1/20 0.41
KMO O15229 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8103529 0.87 AGTR1 (0.44) AGTR1AGTR2ALOX5APNPC1RAB9A
SCHEMBL8111149 0.85 PPARG (0.49) PPARGALOX5APPDE7APDE7BNPC1
SCHEMBL8109337 0.85 PPARG (0.47) AGTR1AGTR2PPARGALOX5APPDE7A
SCHEMBL8105380 0.82 PPARG (0.62) AGTR1AGTR2PPARGNPC1RAB9A
SCHEMBL8103387 0.81 PPARG (0.50) AGTR1AGTR2PPARG
SCHEMBL8105265 0.80 PPARG (0.55) AGTR1AGTR2PPARG
SCHEMBL6005987 0.80 AGTR1 (0.73) AGTR1AGTR2
SCHEMBL8103632 0.79 PPARG (0.49) PPARGPDE7APDE7BNPC1RAB9A
SCHEMBL8103636 0.79 PPARG (0.49) PPARGPDE7APDE7BNPC1RAB9A
SCHEMBL8095962 0.79 PPARG (0.56) AGTR1AGTR2PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3098772-B2 2000-10-16 JP claimed
EP-0527851-A1 1H-SUBSTITUTED-1,2,4-TRIAZOLE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1993-02-24 EP claimed
WO-1991017148-A1 1H-SUBSTITUTED-1,2,4-TRIAZOLE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1991-11-14 WO claimed
EP-0527851-A1 1H-SUBSTITUTED-1,2,4-TRIAZOLE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1993-02-24 EP disclosed
US-5098920-A Hypotensive agents and treatment of congestive heart failure G. D. SEARLE & CO. (US) 1992-03-24 US disclosed
WO-1991017148-A1 1H-SUBSTITUTED-1,2,4-TRIAZOLE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1991-11-14 WO disclosed