SCHEMBL8111149

SCHEMBL8111149

CC(C)CCc1nc(CCC(C)C)n(Cc2ccc(-c3cccc(C(=O)O)c3)cc2)n1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.49
PDE7A Q13946 1/20 0.42
PDE7B Q9NP56 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ALOX5AP P20292 1/20 0.42
MGLL Q99685 1/20 0.40
DHFR P00374 1/20 0.40
MAP1LC3B Q9GZQ8 1/20 0.40
MAP1LC3A Q9H492 1/20 0.40
HDAC6 Q9UBN7 1/20 0.39
KMO O15229 1/20 0.39
ADRB3 P13945 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8103387 0.93 PPARG (0.50) PPARG
SCHEMBL8103506 0.88 CA1 (0.39) PPARGNPC1RAB9ASMN1; SMN2
SCHEMBL8105380 0.86 PPARG (0.62) PPARGNPC1RAB9ASMN1; SMN2DHFR
SCHEMBL8111214 0.86 PPARG (0.49) PPARGPDE7APDE7BNPC1RAB9A
SCHEMBL8096036 0.85 AGTR1 (0.48) PPARGPDE7APDE7BNPC1RAB9A
SCHEMBL8105265 0.84 PPARG (0.55) PPARG
SCHEMBL8096101 0.84 PPARG (0.54) PPARG
SCHEMBL8104965 0.84 PPARG (0.59) PPARG
SCHEMBL8095962 0.84 PPARG (0.56) PPARG
SCHEMBL8095655 0.82 AGTR1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3098772-B2 2000-10-16 JP claimed
EP-0527851-A1 1H-SUBSTITUTED-1,2,4-TRIAZOLE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1993-02-24 EP claimed
WO-1991017148-A1 1H-SUBSTITUTED-1,2,4-TRIAZOLE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1991-11-14 WO claimed
EP-0527851-A1 1H-SUBSTITUTED-1,2,4-TRIAZOLE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1993-02-24 EP disclosed
US-5098920-A Hypotensive agents and treatment of congestive heart failure G. D. SEARLE & CO. (US) 1992-03-24 US disclosed
WO-1991017148-A1 1H-SUBSTITUTED-1,2,4-TRIAZOLE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1991-11-14 WO disclosed