SCHEMBL8096598

SCHEMBL8096598

CC(C)N(C(=O)CC(C#N)c1ccccc1)C(C)C.CC(C)N(C(=O)CC(C(N)=O)c1ccccc1)C(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.41
ALOX5 P09917 1/20 0.38
TRPM8 Q7Z2W7 2/20 0.36
KCNA5 P22460 1/20 0.36
ALDH1A1 P00352 3/20 0.35
TDP1 Q9NUW8 1/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
GAA P10253 1/20 0.34
AKR1C3 P42330 1/20 0.34
AKR1C1 Q04828 1/20 0.34
LMNA P02545 2/20 0.34
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MMP9 P14780 1/20 0.33
MMP8 P22894 1/20 0.33
MMP13 P45452 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6934985 0.89 KCNA5 (0.42) ALOX5KCNA5ALDH1A1KMT2AMEN1
SCHEMBL6937352 0.88 EPHX1 (0.51) EPHX1ALOX5TRPM8KCNA5ALDH1A1
SCHEMBL6063192 0.73 CYP2C19 (0.47) EPHX1ALOX5ALDH1A1TDP1KMT2A
SCHEMBL6798718 0.73 CYP2C19 (0.47) EPHX1ALOX5ALDH1A1TDP1KMT2A
SCHEMBL6939334 0.72 MMP8 (0.47) KCNA5ALDH1A1KMT2AMEN1GAA
SCHEMBL12718845 0.71 EPHX1 (0.59) EPHX1ALOX5ALDH1A1LMNAKDM4E
SCHEMBL11568787 0.70 KMT2A (0.46) ALDH1A1TDP1KMT2AMEN1AKR1C3
SCHEMBL1343883 0.70 FFAR1 (0.51) KMT2A
SCHEMBL9556420 0.70 FFAR1 (0.51) KMT2A
SCHEMBL27862777 0.70 FFAR1 (0.51) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1019358-A1 NOVEL COMPOUNDS, THEIR USE AND PREPARATION Pharmacia & Upjohn AB (SE) 2000-07-19 EP disclosed
WO-1998043942-A1 NOVEL COMPOUNDS, THEIR USE AND PREPARATION PHARMACIA & UPJOHN AB (SE) 1998-10-08 WO disclosed