SCHEMBL8096733

SCHEMBL8096733

COC(=O)C=C1C2CC3CC1CC(c1ccccc1)(C3)C2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.39
HIF1A Q16665 4/20 0.38
EPAS1 Q99814 2/20 0.38
HSD11B1 P28845 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
SLC6A3 Q01959 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
EPHX2 P34913 1/20 0.38
RAB9A P51151 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RCE1 Q9Y256 1/20 0.36
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8096982 0.76 TSHR (0.37) HSD11B1EPHX2
SCHEMBL8799889 0.75 TSHR (0.36) HSD11B1EPHX2NPSR1
SCHEMBL1397580 0.72 GRIN2D (0.46) LMNANPC1ALDH1A1HSD11B1MEN1
SCHEMBL2749102 0.71 TSHR (0.59) NPC1ALDH1A1SLC6A3MEN1KMT2A
SCHEMBL29319319 0.69 MEN1 (0.42) LMNAALDH1A1HSD11B1SIGMAR1MEN1
SCHEMBL181479 0.69 GRIN2D (0.62) LMNANPC1ALDH1A1HSD11B1MEN1
SCHEMBL19174005 0.69 GRIN2D (0.46) LMNANPC1ALDH1A1HSD11B1MEN1
SCHEMBL8097125 0.68 LMNA (0.45) LMNANPC1HIF1AEPAS1HSD11B1
Acetanilide SCHEMBL29173779 0.68 NPC1 (0.80) LMNANPC1ALDH1A1KMT2AEPHX2
SCHEMBL23567005 0.67 S1PR5 (0.46) LMNASIGMAR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0661271-B1 AZEPINE DERIVATIVES, PRODUCTION THEREOF, AND USE THEREOF AS SIGMA-RECEPTOR LIGANDS ASAHI CHEMICAL IND (JP) 2000-04-26 EP disclosed
US-5658923-A USED IN TREATING DISEASES RELATED TO SIGMA-RECEPTOR, SUCH AS SCHIZOPHRENIA ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1997-08-19 US disclosed
EP-0661271-A1 AZEPINE DERIVATIVE, PRODUCTION THEREOF, AND USE THEREOF Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1995-07-05 EP disclosed