SCHEMBL8097062

SCHEMBL8097062

COC(=O)[C@@H]1C[C@H](C(=O)NC(C)(Cc2ccc(C#N)cc2)c2cnc[nH]2)CN(CC(c2ccccc2)c2ccccc2)C1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 6/20 0.36
CCR5 P51681 3/20 0.34
EP300 Q09472 5/20 0.33
FNTA P49354 5/20 0.33
FNTB P49356 5/20 0.33
LTA4H P09960 1/20 0.31
HAT1 O14929 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8097065 1.00 CYP19A1 (0.36) CYP19A1CCR5EP300FNTAFNTB
SCHEMBL8103769 1.00 CYP19A1 (0.36) CYP19A1CCR5EP300FNTAFNTB
SCHEMBL8097890 0.93 CYP19A1 (0.37) CYP19A1CCR5EP300FNTAFNTB
SCHEMBL8097886 0.93 CYP19A1 (0.37) CYP19A1CCR5EP300FNTAFNTB
SCHEMBL8098343 0.91 HRH3 (0.33) CYP19A1FNTAFNTB
SCHEMBL8098346 0.91 HRH3 (0.33) CYP19A1FNTAFNTB
SCHEMBL8095949 0.90 FNTA (0.37) FNTAFNTB
SCHEMBL8095942 0.90 FNTA (0.37) FNTAFNTB
SCHEMBL8101922 0.89 CYP19A1 (0.34) CYP19A1CCR5EP300FNTAFNTB
SCHEMBL8101919 0.89 CYP19A1 (0.34) CYP19A1CCR5EP300FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127366-A ANTICARCINOGENIC OR ANTITUMOR AGENTS MERCK & CO., INC. (US) 2000-10-03 US disclosed
US-5817678-A IMIDAZOLE-CONTAINING PIPERIDINE DERIVATIVES, PEPTIDEMIMETIC MERCK & CO., INC. (US) 1998-10-06 US disclosed