SCHEMBL8097174

SCHEMBL8097174

CC(=O)NCCOc1ccc(Cl)c(COc2ccc3nc(C)ccc3c2)c1Cl

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 7/20 0.40
KLKB1 P03952 2/20 0.40
S1PR4 O95977 1/20 0.39
RAB9A P51151 1/20 0.39
PPARG P37231 1/20 0.39
SCN9A Q15858 1/20 0.39
MTNR1A P48039 2/20 0.37
MTNR1B P49286 2/20 0.37
NCF1 P14598 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
ACSS2 Q9NR19 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8099739 0.85 BDKRB2 (0.42) BDKRB2KLKB1RAB9APPARGMTNR1A
SCHEMBL8098950 0.83 S1PR4 (0.37) BDKRB2KLKB1S1PR4PPARGNCF1
SCHEMBL8097169 0.80 BDKRB2 (0.60) BDKRB2
SCHEMBL8106164 0.77 HPGD (0.44) KLKB1RAB9AALDH1A1HPGD
SCHEMBL6936592 0.75 KDM4E (0.42) RAB9ANCF1KDM4EALDH1A1
SCHEMBL6581385 0.73 TP53 (0.42) S1PR4ALDH1A1HPGD
SCHEMBL6935565 0.72 BDKRB2 (0.46) BDKRB2
SCHEMBL8105709 0.70 BDKRB2 (0.57) BDKRB2
SCHEMBL8098918 0.70 BDKRB2 (0.60) BDKRB2
SCHEMBL8090589 0.69 BDKRB2 (0.59) BDKRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795547-B1 (Aminoalkyl- and acylaminoalkyl-oxy)benzyloxyquinolines, process for their preparation and use as Bradykinin receptor antagonists HOECHST AG (DE) 2000-05-10 EP claimed