SCHEMBL8098378

SCHEMBL8098378

COC(=O)[C@@H]1C[C@H](C(=O)NC(C)(Cc2ccc(C#N)cc2)c2cnc[nH]2)CN(C)C1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 3/20 0.34
CYP11B2 P19099 3/20 0.34
HRH3 Q9Y5N1 1/20 0.33
FNTA P49354 2/20 0.33
FNTB P49356 2/20 0.33
GPR119 Q8TDV5 1/20 0.33
DPP4 P27487 1/20 0.32
ACACB O00763 1/20 0.32
GPBAR1 Q8TDU6 3/20 0.31
ERG P11308 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP19A1 P11511 1/20 0.31
KDM1A O60341 1/20 0.31
CTSS P25774 1/20 0.31
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC4 P56524 1/20 0.30
HDAC1 Q13547 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8098386 1.00 CYP11B1 (0.34) CYP11B1CYP11B2HRH3FNTAFNTB
SCHEMBL8444117 0.90 GPR119 (0.42) CYP11B1CYP11B2GPR119ACACB
SCHEMBL8097497 0.90 GPR119 (0.42) CYP11B1CYP11B2GPR119ACACB
SCHEMBL8098346 0.90 HRH3 (0.33) CYP11B1CYP11B2HRH3FNTAFNTB
SCHEMBL8098343 0.90 HRH3 (0.33) CYP11B1CYP11B2HRH3FNTAFNTB
SCHEMBL8097494 0.90 GPR119 (0.42) CYP11B1CYP11B2GPR119ACACB
SCHEMBL8096857 0.90 GPR119 (0.42) CYP11B1CYP11B2GPR119ACACB
SCHEMBL8097913 0.89 L3MBTL1 (0.39) HRH3FNTAFNTBCYP19A1L3MBTL1
SCHEMBL8097906 0.89 L3MBTL1 (0.39) HRH3FNTAFNTBCYP19A1L3MBTL1
SCHEMBL8097797 0.89 CHRM4 (0.35) CYP11B1CYP11B2HRH3FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127366-A ANTICARCINOGENIC OR ANTITUMOR AGENTS MERCK & CO., INC. (US) 2000-10-03 US disclosed
US-5817678-A IMIDAZOLE-CONTAINING PIPERIDINE DERIVATIVES, PEPTIDEMIMETIC MERCK & CO., INC. (US) 1998-10-06 US disclosed