SCHEMBL8098384

SCHEMBL8098384

CC(C[C@@H]1C[C@@H](O[Si](C)(C)C(C)(C)C)CN1C(=O)OC(C)(C)C)N1C(=O)c2ccccc2C1=O

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.38
IDO1 P14902 4/20 0.37
SRC P12931 7/20 0.35
PARP1 P09874 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
UCHL1 P09936 1/20 0.33
HTRA1 Q92743 1/20 0.33
KLK7 P49862 1/20 0.33
KLK5 Q9Y337 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
USP2 O75604 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3948504 0.85 ABCB1 (0.38) ABCB1IDO1SRCPARP1UCHL1
SCHEMBL21286395 0.85 ABCB1 (0.38) ABCB1IDO1SRCPARP1UCHL1
SCHEMBL29985450 0.85 ABCB1 (0.38) ABCB1IDO1SRCPARP1UCHL1
SCHEMBL1526220 0.83 ABCB1 (0.37) ABCB1IDO1SRCPARP1UCHL1
SCHEMBL1526218 0.83 ABCB1 (0.37) ABCB1IDO1SRCPARP1UCHL1
SCHEMBL8106554 0.81 ABCB1 (0.35) ABCB1IDO1SRCPARP1HTRA1
SCHEMBL9595418 0.81 ABCB1 (0.35) ABCB1IDO1SRCPARP1HTRA1
SCHEMBL7859886 0.78 NR1H2 (0.46) ABCB1SRCPARP1UCHL1KLK7
SCHEMBL8107520 0.78 NR1H2 (0.34) ABCB1SRC
SCHEMBL3948290 0.77 ABCB1 (0.41) ABCB1SRCPARP1UCHL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0545290-B1 Aminoalkylpyrrolidinylthiocarbapenem derivatives BANYU PHARMA CO LTD (JP) 2000-08-23 EP disclosed
US-5550121-A ANTIBIOTICS BANYU PHARMACEUTICAL CO., LTD. (JP) 1996-08-27 US disclosed
WO-1993011128-A1 AMINOALKYLPYRROLIDINYLTHIOCARBAPENEM DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-06-10 WO disclosed
EP-0545290-A1 Aminoalkylpyrrolidinylthiocarbapenem derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-06-09 EP disclosed