SCHEMBL8098696

SCHEMBL8098696

CCCCOc1nc(-c2ccc(SC)cc2)c(-c2ccc(S(N)(=O)=O)cc2)cc1C#N

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.47
PTGS1 P23219 5/20 0.47
CA2 P00918 5/20 0.42
CNR1 P21554 4/20 0.42
CA1 P00915 4/20 0.42
CA7 P43166 4/20 0.42
CA12 O43570 3/20 0.42
CA9 Q16790 3/20 0.42
TSHR P16473 1/20 0.42
CDK1 P06493 1/20 0.38
KDR P35968 1/20 0.38
CHUK O15111 2/20 0.38
IKBKB O14920 1/20 0.37
CA13 Q8N1Q1 1/20 0.37
CA14 Q9ULX7 1/20 0.37
TTK P33981 1/20 0.36
MAPK8 P45983 1/20 0.36
CA5A P35218 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8086268 0.91 PTGS2 (0.57) PTGS2PTGS1CNR1CHUKIKBKB
SCHEMBL8094646 0.91 PTGS2 (0.42) PTGS2PTGS1CA2CNR1CA1
SCHEMBL8087099 0.90 PTGS2 (0.48) PTGS2PTGS1CA2CNR1CA1
SCHEMBL8094547 0.89 PTGS2 (0.60) PTGS2PTGS1CA2CNR1CA1
SCHEMBL8095632 0.86 PTGS2 (0.56) PTGS2PTGS1CA2CNR1CA1
SCHEMBL8093748 0.86 KDM4E (0.43) PTGS2PTGS1CA2CNR1CA1
SCHEMBL8092530 0.86 PTGS2 (0.55) PTGS2PTGS1CA2CNR1CA1
SCHEMBL8095681 0.85 CA2 (0.51) PTGS2PTGS1CA2CNR1CA1
SCHEMBL8086798 0.85 PTGS2 (0.44) PTGS2PTGS1CA2CNR1CA1
SCHEMBL8095136 0.84 PTGS2 (0.66) PTGS2PTGS1CA2CNR1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed