SCHEMBL8098772

SCHEMBL8098772

CCCNC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4nc(C)cs4)CC3)n2)cc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 8/20 0.39
PIK3CA P42336 6/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
RAB9A P51151 1/20 0.36
KDR P35968 2/20 0.36
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
GHSR Q92847 1/20 0.35
MTOR P42345 2/20 0.34
KIT P10721 1/20 0.34
MMP2 P08253 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
PIK3CG P48736 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8089088 0.93 PIK3CA (0.40) PIK3CDPIK3CARAB9AKDRMTOR
SCHEMBL8096194 0.92 KDM4E (0.39) PIK3CDPIK3CARAB9AKDRMTOR
SCHEMBL8085149 0.90 PIK3CA (0.39) PIK3CDPIK3CARAB9AKDRMTOR
SCHEMBL8090804 0.89 MTOR (0.37) PIK3CDPIK3CARAB9AKDRMTOR
SCHEMBL8097960 0.89 KDM4E (0.38) PIK3CDPIK3CARAB9AKDRMTOR
SCHEMBL8091977 0.86 PIK3CD (0.35) PIK3CDPIK3CARAB9A
SCHEMBL8096192 0.85 PIK3CD (0.36) PIK3CDPIK3CARAB9AKDRMTOR
SCHEMBL3928570 0.85 PIK3CA (0.52) PIK3CDPIK3CAMTORPIK3CG
SCHEMBL8089090 0.85 KDR (0.39) PIK3CARAB9AKDRMTORKIT
SCHEMBL8092385 0.84 PIK3CD (0.41) PIK3CDPIK3CAKDRGHSRMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed