SCHEMBL8099890

SCHEMBL8099890

CC(C)NC(=O)Nc1ccc(-c2nc(N)cc(C3(SO)CC3)n2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 1/20 0.39
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA9 Q16790 2/20 0.39
ROCK2 O75116 4/20 0.39
CYP3A4 P08684 2/20 0.37
CYP3A5 P20815 2/20 0.37
LIMK1 P53667 4/20 0.36
MEN1 O00255 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 2/20 0.36
HPGD P15428 2/20 0.36
KMT2A Q03164 2/20 0.36
RXFP1 Q9HBX9 2/20 0.36
KDM4E B2RXH2 1/20 0.36
EPHX2 P34913 1/20 0.36
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8095224 0.90 PIK3CD (0.34) GHSRCA12CA1CA2CA9
SCHEMBL8090988 0.88 MTOR (0.44) MEN1ALDH1A1MAPTHPGDKMT2A
SCHEMBL8089937 0.85 KIF11 (0.39) MEN1ALDH1A1MAPTHPGDKMT2A
SCHEMBL8095600 0.82 CA12 (0.39) GHSRCA12CA1CA2CA9
SCHEMBL8098188 0.82 CA12 (0.44) GHSRCA12CA1CA2CA9
SCHEMBL8091600 0.82 PIK3CA (0.40) PIK3CD
SCHEMBL8089531 0.82 CA12 (0.43) GHSRCA12CA1CA2CA9
SCHEMBL8083982 0.82 PIK3CD (0.34) MEN1ALDH1A1MAPTHPGDKMT2A
SCHEMBL8097252 0.82 CA12 (0.43) GHSRCA12CA1CA2CA9
SCHEMBL8091781 0.82 CA12 (0.43) GHSRCA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed