SCHEMBL8100548

SCHEMBL8100548

N#Cc1cc(-c2ccc(S(N)(=O)=O)cc2)c(-c2ccc(F)cc2)nc1SCC1CCCCC1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.44
PTGS1 P23219 7/20 0.44
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
DPP4 P27487 1/20 0.40
CA12 O43570 3/20 0.40
CA1 P00915 3/20 0.40
CA2 P00918 3/20 0.40
CA9 Q16790 3/20 0.40
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
IKBKB O14920 1/20 0.36
CHUK O15111 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8095856 0.99 ALDH1A1 (0.43) PTGS2PTGS1ALDH1A1LMNADPP4
SCHEMBL8094759 0.91 PTGS2 (0.55) PTGS2PTGS1ALDH1A1LMNA
SCHEMBL8099590 0.90 PTGS2 (0.54) PTGS2PTGS1ALDH1A1LMNA
SCHEMBL8776719 0.89 PTGS2 (0.44) PTGS2PTGS1ALDH1A1LMNACNR1
SCHEMBL8094910 0.83 PTGS2 (0.46) PTGS2PTGS1CNR1CNR2
SCHEMBL8094996 0.83 PTGS2 (0.48) PTGS2PTGS1DPP4CA12CA1
SCHEMBL8094384 0.82 MAPK13 (0.47) PTGS2PTGS1ALDH1A1LMNACA12
SCHEMBL8101167 0.82 PTGS2 (0.45) PTGS2PTGS1CNR1CNR2IKBKB
SCHEMBL8093245 0.81 ALDH1A1 (0.45) PTGS2PTGS1ALDH1A1LMNACA12
SCHEMBL8098730 0.80 CNR1 (0.44) PTGS2PTGS1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed