SCHEMBL8776719

SCHEMBL8776719

CCS(=O)(=O)c1ccc(-c2cc(C#N)c(SCC3CCCC3)nc2-c2ccc(F)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.44
PTGS1 P23219 5/20 0.44
ALDH1A1 P00352 2/20 0.43
LMNA P02545 1/20 0.43
RORC P51449 3/20 0.38
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
MAPK13 O15264 1/20 0.35
MAPK12 P53778 1/20 0.35
MAPK11 Q15759 1/20 0.35
MAPK14 Q16539 1/20 0.35
GABRA2 P47869 1/20 0.35
KDM1A O60341 1/20 0.35
AR P10275 2/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8099590 0.92 PTGS2 (0.54) PTGS2PTGS1ALDH1A1LMNAMAPK13
SCHEMBL8094759 0.91 PTGS2 (0.55) PTGS2PTGS1ALDH1A1LMNAMAPK13
SCHEMBL8095856 0.90 ALDH1A1 (0.43) PTGS2PTGS1ALDH1A1LMNACNR1
SCHEMBL8100548 0.89 PTGS2 (0.44) PTGS2PTGS1ALDH1A1LMNACNR1
SCHEMBL8776749 0.78 PTGS2 (0.47) PTGS2PTGS1ALDH1A1LMNARORC
SCHEMBL8420124 0.76 ALDH1A1 (0.39) PTGS2PTGS1ALDH1A1LMNANPSR1
SCHEMBL8776720 0.76 PTGS2 (0.47) PTGS2PTGS1CNR1CNR2L3MBTL1
SCHEMBL8776825 0.76 PTGS2 (0.46) PTGS2PTGS1ALDH1A1RORCCNR1
SCHEMBL8420193 0.76 MCL1 (0.39) PTGS2PTGS1ALDH1A1LMNANPSR1
SCHEMBL8101431 0.75 PTGS2 (0.56) PTGS2PTGS1CNR1CNR2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed