SCHEMBL8101985

SCHEMBL8101985

Cc1ccc2nc(-c3cccc4ccccc34)cc(=O)n2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 2/20 0.46
GRIN2A Q12879 2/20 0.46
PARP1 P09874 1/20 0.45
PKM P14618 3/20 0.44
KDM4E B2RXH2 5/20 0.42
ALDH1A1 P00352 5/20 0.42
HPGD P15428 2/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
FLT3 P36888 1/20 0.42
POLB P06746 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL32688213 0.85 GRIN1 (0.48) GRIN1GRIN2APARP1PKMKDM4E
SCHEMBL8092506 0.82 ALDH1A1 (0.55) PARP1PKMKDM4EALDH1A1HPGD
SCHEMBL8102203 0.81 HSP90AA1 (0.47) PARP1PKMKDM4EALDH1A1HPGD
SCHEMBL7920187 0.81 DCTPP1 (0.48) GRIN1GRIN2APKMKDM4EALDH1A1
SCHEMBL32688343 0.81 DCTPP1 (0.48) GRIN1GRIN2APKMKDM4EALDH1A1
SCHEMBL32688219 0.80 GRIN1 (0.44) GRIN1GRIN2APARP1PKMKDM4E
SCHEMBL1660663 0.79 NPC1 (0.56) GRIN1GRIN2APKMKDM4EALDH1A1
SCHEMBL28615697 0.77 NPC1 (0.58) PKMKDM4EALDH1A1HPGDTSHR
SCHEMBL8099857 0.77 NR1H4 (0.50) GRIN1GRIN2APARP1PKMKDM4E
SCHEMBL8099803 0.77 NPC1 (0.51) GRIN1GRIN2APKMKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6071930-A FOR INHIBITION OF MITOSIS OR TUMOR GROWTH THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2000-06-06 US disclosed
US-5994367-A PREVENT CELL MITOSIS; ANTICARCINOGENIC AGENTS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1999-11-30 US disclosed