SCHEMBL8102006

SCHEMBL8102006

Cc1cccc2nc(-c3ccc(F)cc3)cc(=O)n12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.55
GRIN2A Q12879 1/20 0.55
MAPT P10636 3/20 0.49
TP53 P04637 2/20 0.49
THRB P10828 1/20 0.49
RAD51 Q06609 4/20 0.49
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 3/20 0.45
HPGD P15428 2/20 0.45
KDM5B Q9UGL1 1/20 0.44
CYP1A2 P05177 1/20 0.43
POLB P06746 1/20 0.43
CYP2C19 P33261 1/20 0.43
CDC7 O00311 1/20 0.43
PIM1 P11309 1/20 0.43
GSK3B P49841 1/20 0.43
HIPK2 Q9H2X6 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
PSD A5PKW4 2/20 0.43
NPC1 O15118 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8106228 0.88 RAD51 (0.54) GRIN1GRIN2AMAPTTP53RAD51
SCHEMBL4440840 0.87 GRIN1 (0.51) GRIN1GRIN2AMAPTTP53THRB
SCHEMBL1537159 0.87 KDM4E (0.55) GRIN1GRIN2ATP53RAD51ALDH1A1
SCHEMBL8101357 0.86 HTT (0.49) MAPTTP53RAD51ALDH1A1KDM4E
SCHEMBL7921851 0.83 PKM (0.49) MAPTTP53ALDH1A1KDM4EHPGD
SCHEMBL8100020 0.83 RAD51 (0.49) MAPTTP53THRBRAD51ALDH1A1
SCHEMBL8102003 0.82 PKM (0.44) GRIN1GRIN2ARAD51ALDH1A1KDM4E
SCHEMBL8101399 0.81 NPC1 (0.52) GRIN1GRIN2AMAPTRAD51ALDH1A1
SCHEMBL8108081 0.79 GAA (0.50) GRIN1GRIN2AMAPTTP53RAD51
SCHEMBL8106086 0.77 MEN1 (0.54) MAPTTP53ALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6071930-A FOR INHIBITION OF MITOSIS OR TUMOR GROWTH THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2000-06-06 US disclosed
US-5994367-A PREVENT CELL MITOSIS; ANTICARCINOGENIC AGENTS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1999-11-30 US disclosed