SCHEMBL8102003

SCHEMBL8102003

Cc1cccc2nc(-c3ccc4ccccc4c3)cc(=O)n12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.44
CTRC Q99895 1/20 0.43
CYP1A2 P05177 2/20 0.42
HTT P42858 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
RAD51 Q06609 3/20 0.41
KDM4E B2RXH2 2/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
CYP1A1 P04798 1/20 0.40
CYP1B1 Q16678 1/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
RAC1 P63000 2/20 0.39
GSTP1 P09211 1/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1537159 0.85 KDM4E (0.55) PKMCYP1A2HTTRXFP1RAD51
SCHEMBL8106201 0.85 CTRC (0.45) CTRCCYP1A2RAD51KDM4ENPC1
SCHEMBL8106228 0.84 RAD51 (0.54) PKMCYP1A2HTTRXFP1RAD51
SCHEMBL8101399 0.83 NPC1 (0.52) PKMCYP1A2HTTRXFP1RAD51
SCHEMBL7921851 0.82 PKM (0.49) PKMKDM4ENPC1RAB9AALDH1A1
SCHEMBL8101357 0.82 HTT (0.49) PKMHTTRXFP1RAD51KDM4E
SCHEMBL8102006 0.82 GRIN1 (0.55) PKMCYP1A2HTTRXFP1RAD51
SCHEMBL8106086 0.81 MEN1 (0.54) RXFP1KDM4ENPC1RAB9AALDH1A1
SCHEMBL8108081 0.81 GAA (0.50) PKMCYP1A2HTTRXFP1RAD51
SCHEMBL4440840 0.81 GRIN1 (0.51) PKMCYP1A2HTTRXFP1RAD51

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6071930-A FOR INHIBITION OF MITOSIS OR TUMOR GROWTH THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2000-06-06 US disclosed
US-5994367-A PREVENT CELL MITOSIS; ANTICARCINOGENIC AGENTS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1999-11-30 US disclosed