SCHEMBL8102527

SCHEMBL8102527

COc1ccc(C(C#N)C(O)C2CCCCC2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.58
SLC6A4 P31645 2/20 0.58
SLC6A3 Q01959 2/20 0.58
CHRM2 P08172 7/20 0.44
CHRM1 P11229 7/20 0.44
CHRM4 P08173 5/20 0.44
CHRM3 P20309 4/20 0.44
CHRM5 P08912 1/20 0.43
EPHX2 P34913 1/20 0.42
ALDH1A1 P00352 3/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
MAPT P10636 2/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4246228 0.77 CHRM2 (0.60) SLC6A2SLC6A4SLC6A3CHRM2CHRM1
SCHEMBL4611536 0.77 SLC6A2 (0.60) SLC6A2SLC6A4SLC6A3CHRM2CHRM1
SCHEMBL4996406 0.76 SLC6A3 (0.56) SLC6A2SLC6A4SLC6A3MEN1KMT2A
SCHEMBL14115528 0.76 SLC6A3 (0.56) SLC6A2SLC6A4SLC6A3MEN1KMT2A
SCHEMBL20970365 0.75 SLC6A2 (0.75) SLC6A2SLC6A4SLC6A3EPHX2ALDH1A1
SCHEMBL1095179 0.75 ALDH1A1 (0.49) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
Hydrochloric Acid SCHEMBL8110122 0.73 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3EPHX2ALDH1A1
SCHEMBL25620291 0.73 SLC6A2 (0.55) SLC6A2SLC6A4SLC6A3CHRM2CHRM1
SCHEMBL12551531 0.72 ESR2 (0.70) ALDH1A1MEN1KMT2AMAPTCYP3A4
Hydrochloric Acid SCHEMBL8116973 0.71 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3EPHX2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6069177-A ADMINISTERING TO THE HUMAN AN EFFECTIVE ANTIDEPRESSANT DOSE OF THE COMPOUND 3-HYDROXY-4,4-DIMETHYL-2-(2'-NAPHTHYL)PENTYL-N,N-DIMETHYLAMINE OR SALT THE HONG KONG UNIVERSITY OF SCIENCE AND TECHNOLOGY (HK) 2000-05-30 US disclosed