SCHEMBL8103025

SCHEMBL8103025

CNCC(=O)Nc1ccc2ncnc(Nc3ccc(F)c(F)c3)c2c1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.61
AURKB Q96GD4 2/20 0.61
ERBB2 P04626 5/20 0.56
ERBB4 Q15303 1/20 0.56
HDAC6 Q9UBN7 2/20 0.55
HDAC1 Q13547 1/20 0.55
FYN P06241 1/20 0.55
GMPS P49915 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8104687 0.86 EGFR (0.70) EGFRAURKBERBB2ERBB4HDAC6
SCHEMBL8104967 0.81 EGFR (0.57) EGFRERBB2ERBB4
SCHEMBL8110759 0.79 EGFR (0.74) EGFRERBB2ERBB4
SCHEMBL2248477 0.77 EGFR (0.77) EGFRAURKBERBB2ERBB4HDAC6
SCHEMBL27819297 0.77 EGFR (0.74) EGFRAURKBERBB2ERBB4HDAC6
SCHEMBL7763004 0.76 ALK (0.60) EGFRERBB2
SCHEMBL7766632 0.76 EGFR (0.57) EGFRERBB2ERBB4HDAC6HDAC1
SCHEMBL8310027 0.76 EGFR (0.66) EGFRAURKBERBB2ERBB4GMPS
SCHEMBL2255586 0.75 EGFR (0.74) EGFRAURKBERBB2ERBB4HDAC6
SCHEMBL7760716 0.75 EGFR (0.70) EGFRAURKBERBB2ERBB4HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6015814-A Quinazoline derivative ZENECA LIMITED (GB) 2000-01-18 US disclosed
EP-0824526-A1 QUINAZOLINE DERIVATIVE ZENECA LIMITED (GB) 1998-02-25 EP disclosed
WO-1996033978-A1 QUINAZOLINE DERIVATIVE ZENECA LIMITED (GB) 1996-10-31 WO disclosed