SCHEMBL8103205

SCHEMBL8103205

COc1cc(OC)c(C(F)(F)F)cc1C(=O)NC(=N)N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 6/20 0.40
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
SLC9A1 P19634 1/20 0.37
CFTR P13569 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LRRK2 Q5S007 1/20 0.36
CYP2C9 P11712 2/20 0.35
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPK8 P45983 1/20 0.35
MAPK10 P53779 1/20 0.35
CYP1A2 P05177 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8117208 0.99 S1PR1 (0.39) S1PR1HTR2AHTR2CSLC9A1CFTR
Hydrochloric Acid SCHEMBL7805318 0.90 TNFSF11 (0.40) S1PR1SLC9A1ALDH1A1LRRK2CYP2C9
SCHEMBL7801887 0.89 APP (0.39) S1PR1SLC9A1CFTRLRRK2CYP2C9
SCHEMBL8428710 0.88 MAPT (0.40) S1PR1HTR2AHTR2CLRRK2MAPT
Hydrochloric Acid SCHEMBL8335173 0.87 MAPT (0.40) S1PR1HTR2AHTR2CLRRK2MAPT
SCHEMBL8116932 0.80 MAPT (0.47) CFTRMAPTKDM4E
Hydrochloric Acid SCHEMBL8102752 0.78 MAPT (0.46) CFTRMAPT
SCHEMBL8102763 0.77 CFTR (0.49) HTR2AHTR2CCFTRALDH1A1MAPT
SCHEMBL1763883 0.77 SLC9A1 (0.69) HTR2ASLC9A1CYP2C9CYP2C19
SCHEMBL5874056 0.76 ALDH1A1 (0.50) HTR2AHTR2CALDH1A1KDM4ECYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153651-A Ortho-substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament comprising them HOECHST AKTIENGESELLSCHAFT (DE) 2000-11-28 US claimed