SCHEMBL8103240

SCHEMBL8103240

O=CC1(Cc2ccccn2)CN(C(=O)O)CCN1C(=O)OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 6/20 0.41
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 3/20 0.40
GRM5 P41594 1/20 0.40
POLB P06746 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
CYP2C19 P33261 1/20 0.36
F13A1 P00488 1/20 0.36
TGM2 P21980 1/20 0.36
TGM1 P22735 1/20 0.36
CYP2D6 P10635 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5228286 0.89 MEN1 (0.42) GRIN2BKDM4EALDH1A1GRM5POLB
SCHEMBL5227957 0.80 MEN1 (0.40) GRIN2BKDM4EALDH1A1GRM5POLB
SCHEMBL5229398 0.72 MEN1 (0.43) GRIN2BKDM4EALDH1A1POLBMEN1
SCHEMBL17485677 0.71 KDM4E (0.74) GRIN2BKDM4EALDH1A1MEN1KMT2A
SCHEMBL22213481 0.68 CYP2C19 (0.43) MEN1KMT2ANPSR1SMN1; SMN2CYP2C19
SCHEMBL3795583 0.68 MEN1 (0.69) GRIN2BALDH1A1MEN1KMT2ANPSR1
SCHEMBL10333902 0.66
SCHEMBL16611992 0.66 KMT2A (0.67) GRIN2BALDH1A1MEN1KMT2ANPSR1
SCHEMBL3970912 0.66 MEN1 (0.76) GRIN2BALDH1A1MEN1KMT2ANPSR1
SCHEMBL4814264 0.66 MEN1 (0.76) GRIN2BALDH1A1MEN1KMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001970-A1 DIPEPTIDE DERIVATIVES AS GROWTH HORMONE SECRETAGOGUES PFIZER INC. (US) 2000-05-24 EP disclosed
WO-1998058947-A1 DIPEPTIDE DERIVATIVES AS GROWTH HORMONE SECRETAGOGUES PFIZER INC. (US) 1998-12-30 WO disclosed