SCHEMBL8103582

SCHEMBL8103582

C[C@H](NC(=O)C1CCCN(S(=O)(=O)Cc2ccccc2)C1)c1cncn1Cc1ccc(C#N)cc1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.50
LMNA P02545 3/20 0.46
MAPT P10636 2/20 0.46
MEN1 O00255 1/20 0.46
HTT P42858 1/20 0.46
KMT2A Q03164 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ALOX12 P18054 1/20 0.46
HSD17B10 Q99714 1/20 0.45
FNTA P49354 7/20 0.43
FNTB P49356 7/20 0.43
PGGT1B P53609 6/20 0.43
KCNH2 Q12809 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104384 1.00 ALDH1A1 (0.50) ALDH1A1LMNAMAPTMEN1HTT
SCHEMBL8101510 0.91 ALOX12 (0.49) ALDH1A1LMNAMEN1KMT2ASMN1; SMN2
SCHEMBL8097860 0.90 TSHR (0.48) ALDH1A1LMNAKMT2AALOX12FNTA
SCHEMBL8105132 0.86 ALDH1A1 (0.46) ALDH1A1MAPTALOX12FNTAFNTB
SCHEMBL8093696 0.86 CNR1 (0.44) ALDH1A1LMNAHTTKMT2ASMN1; SMN2
SCHEMBL8088953 0.85 FNTA (0.45) ALDH1A1LMNAMAPTHTTKMT2A
SCHEMBL8097930 0.85 FNTA (0.46) FNTAFNTBPGGT1BKCNH2
SCHEMBL8103720 0.85 FNTA (0.46) FNTAFNTBPGGT1BKCNH2
SCHEMBL8097915 0.84 FNTA (0.45) ALOX12FNTAFNTBPGGT1BKCNH2
SCHEMBL8098226 0.84 FNTA (0.45) ALOX12FNTAFNTBPGGT1BKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127366-A ANTICARCINOGENIC OR ANTITUMOR AGENTS MERCK & CO., INC. (US) 2000-10-03 US disclosed