SCHEMBL8103653

SCHEMBL8103653

COc1cccc(N=C=O)c1.O=C=Nc1ccc(Cl)c(Cl)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.65
MAPK1 P28482 1/20 0.65
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3A P46098 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43
TAAR1 Q96RJ0 1/20 0.42
MAPT P10636 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
GAA P10253 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CRHR1 P34998 1/20 0.40
LMNA P02545 1/20 0.40
NPC1 O15118 3/20 0.39
RAB9A P51151 2/20 0.39
GSK3B P49841 4/20 0.39
CYP3A4 P08684 2/20 0.38
TRPA1 O75762 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29541540 0.87 HTR3E (0.53) TDP1MAPK1HTR3EHTR3BHTR3A
SCHEMBL23447 0.87 HTR3E (0.53) TDP1MAPK1HTR3EHTR3BHTR3A
SCHEMBL58874 0.80 MAPK1 (1.00) TDP1MAPK1HTR3EHTR3BHTR3A
SCHEMBL29376406 0.80 MAPK1 (1.00) TDP1MAPK1HTR3EHTR3BHTR3A
SCHEMBL8594415 0.80 TDP1 (0.76) TDP1MAPK1HTR3EHTR3BHTR3A
Dimethylamine SCHEMBL11830270 0.77 MAPK1 (0.85) TDP1MAPK1HTR3EHTR3BHTR3A
SCHEMBL8943270 0.77 CYP3A4 (0.50) TDP1MAPK1HTR3EHTR3BHTR3A
O-Xylene SCHEMBL27865799 0.76 MAPK1 (0.76) TDP1MAPK1HTR3EHTR3BHTR3A
SCHEMBL8942897 0.76 TDP1 (0.76) TDP1MAPK1HTR3EHTR3BHTR3A
SCHEMBL7981297 0.76 MAPK1 (0.88) TDP1MAPK1HTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973936-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 2000-01-26 EP disclosed
WO-1998046786-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed