SCHEMBL8103969

SCHEMBL8103969

CCOC(=O)CCCCCCCC(Br)CC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.49
CYP3A4 P08684 2/20 0.49
TSHR P16473 2/20 0.49
ATM Q13315 1/20 0.49
CYP1A2 P05177 1/20 0.48
KMT2A Q03164 3/20 0.47
ALDH1A1 P00352 4/20 0.45
ALOX15 P16050 2/20 0.45
HSD17B10 Q99714 1/20 0.45
DGKA P23743 1/20 0.44
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.42
POLB P06746 1/20 0.41
LMNA P02545 1/20 0.41
USP2 O75604 1/20 0.41
TRPA1 O75762 1/20 0.41
PAM P19021 2/20 0.41
KDM4E B2RXH2 1/20 0.40
DUSP3 P51452 1/20 0.40
NR1I2 O75469 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3050742 0.93 CYP1A2 (0.52) TDP1CYP3A4TSHRATMCYP1A2
SCHEMBL11283053 0.88 CYP1A2 (0.47) TDP1CYP3A4TSHRATMCYP1A2
SCHEMBL20398910 0.88 TSHR (0.56) TDP1CYP3A4TSHRATMCYP1A2
SCHEMBL7522785 0.85 L3MBTL1 (0.49) TDP1CYP3A4TSHRATMCYP1A2
SCHEMBL4864836 0.84 CYP1A2 (0.47) TDP1CYP3A4TSHRATMCYP1A2
SCHEMBL2715956 0.84 CYP1A2 (0.50) TDP1CYP3A4TSHRATMCYP1A2
SCHEMBL15009773 0.84 CYP1A2 (0.50) TDP1CYP3A4TSHRATMCYP1A2
SCHEMBL10578789 0.84 CYP1A2 (0.50) TDP1CYP3A4TSHRATMCYP1A2
SCHEMBL1800630 0.84 L3MBTL1 (0.51) TDP1CYP3A4TSHRATMKMT2A
SCHEMBL31530896 0.83 DGKA (0.61) TDP1CYP3A4TSHRATMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626969-B1 CoA-IT AND PAF INHIBITORS SMITHKLINE BEECHAM CORP (US) 2000-05-24 EP disclosed
US-5663053-A COENZYME A TRANSACYLASE FOR SCREENING SMITHKLINE BEECHAM CORPORATION (US) 1997-09-02 US disclosed
US-5648373-A CoA-IT and PAF inhibitors SMITHKLINE BEECHAM CORPORATION (US) 1997-07-15 US disclosed
EP-0626969-A4 CoA-IT AND PAF INHIBITORS. SMITHKLINE BEECHAM CORP (US) 1995-04-19 EP disclosed
EP-0626969-A1 CoA-IT AND PAF INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1994-12-07 EP disclosed
WO-1993016674-A1 CoA-IT AND PAF INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1993-09-02 WO disclosed