SCHEMBL8103980

SCHEMBL8103980

CS(=O)(=O)Cc1cc(N)nc(-c2ccc(NC(=O)CC(F)(F)F)cc2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 6/20 0.47
MTOR P42345 4/20 0.47
PIK3CD O00329 6/20 0.46
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
KDM4E B2RXH2 2/20 0.40
MAPT P10636 2/20 0.40
HPGD P15428 2/20 0.40
MAP4K4 O95819 1/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA14 Q9ULX7 1/20 0.38
BACE1 P56817 1/20 0.37
POLB P06746 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
CYP3A4 P08684 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8106097 0.90 PIK3CA (0.46) PIK3CAMTORPIK3CDALDH1A1MEN1
SCHEMBL8093349 0.86 PIK3CD (0.48) PIK3CAMTORPIK3CDALDH1A1MEN1
SCHEMBL8101524 0.86 MEN1 (0.54) PIK3CAMTORPIK3CDALDH1A1MEN1
SCHEMBL8109642 0.85 PIK3CA (0.49) PIK3CAMTORPIK3CDALDH1A1MEN1
SCHEMBL8101525 0.84 TP53 (0.51) PIK3CAMTORPIK3CDALDH1A1MEN1
SCHEMBL11925797 0.84 PIK3CA (0.49) PIK3CAMTORPIK3CDALDH1A1MEN1
SCHEMBL8218786 0.84 PIK3CA (0.53) PIK3CAMTORPIK3CDMEN1KMT2A
SCHEMBL8103957 0.83 PIK3CD (0.47) PIK3CAMTORPIK3CDALDH1A1MEN1
SCHEMBL8104034 0.83 MAPT (0.49) PIK3CAMTORPIK3CDALDH1A1MEN1
SCHEMBL8106035 0.83 PTPN1 (0.52) PIK3CAMTORPIK3CDALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007749-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed