SCHEMBL8104515

SCHEMBL8104515

C[SiH2]OC(O[SiH2]C)C(C)(C)[C@H](COS(=O)(=O)c1ccc(C)cc1)c1ccc(NC(C)=O)nc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.40
RAB9A P51151 1/20 0.38
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 2/20 0.34
KMT2A Q03164 1/20 0.34
LPAR2 Q9HBW0 1/20 0.33
GRIN2B Q13224 1/20 0.33
STAT3 P40763 1/20 0.33
PDE4A P27815 1/20 0.33
PKM P14618 2/20 0.32
CYP1A2 P05177 1/20 0.32
GAA P10253 1/20 0.32
PTK2 Q05397 1/20 0.32
LMNA P02545 1/20 0.32
MAPK1 P28482 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5689585 0.80 RAB9A (0.45) SMN1; SMN2RAB9AKDM4EALDH1A1KMT2A
SCHEMBL5689580 0.80 RAB9A (0.45) SMN1; SMN2RAB9AKDM4EALDH1A1KMT2A
SCHEMBL6136724 0.80 RAB9A (0.45) SMN1; SMN2RAB9AKDM4EALDH1A1KMT2A
SCHEMBL4585228 0.77 SMN1; SMN2 (0.39) SMN1; SMN2RAB9AKDM4EALDH1A1KMT2A
SCHEMBL4585225 0.77 SMN1; SMN2 (0.39) SMN1; SMN2RAB9AKDM4EALDH1A1KMT2A
SCHEMBL4585219 0.77 SMN1; SMN2 (0.39) SMN1; SMN2RAB9AKDM4EALDH1A1KMT2A
SCHEMBL5691476 0.69 CYP1A2 (0.55) SMN1; SMN2RAB9AKDM4EALDH1A1KMT2A
SCHEMBL5691469 0.69 CYP1A2 (0.55) SMN1; SMN2RAB9AKDM4EALDH1A1KMT2A
SCHEMBL6136526 0.66 RAB9A (0.45) SMN1; SMN2RAB9AKDM4EALDH1A1KMT2A
SCHEMBL6136518 0.66 RAB9A (0.45) SMN1; SMN2RAB9AKDM4EALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090942-A Process and intermediates for a β3 -adrenergic receptor agonist PFIZER INC. (US) 2000-07-18 US disclosed