SCHEMBL8104864

SCHEMBL8104864

CN(C)CCCNC(CNC(CCN)N1CCCC1)N1CCCC1

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.37
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104652 0.94 TDP1 (0.41) TDP1CYP2C9CYP2C19
SCHEMBL3931824 0.75
SCHEMBL4881270 0.72 HRH3 (0.39)
SCHEMBL8104876 0.71 KEAP1 (0.40)
SCHEMBL6355310 0.65 TDP1 (0.48) TDP1CYP2C9CYP2C19
SCHEMBL6137087 0.62 TDP1 (0.44) TDP1CYP2C9CYP2C19
SCHEMBL152212 0.61 TDP1 (0.44) TDP1CYP2C9CYP2C19
SCHEMBL28208452 0.60 TDP1 (0.42) TDP1CYP2C9CYP2C19
SCHEMBL19968188 0.60 SLC6A2 (0.34)
SCHEMBL28685038 0.59 TDP1 (0.48) TDP1CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6015814-A Quinazoline derivative ZENECA LIMITED (GB) 2000-01-18 US claimed
US-6015814-A Quinazoline derivative ZENECA LIMITED (GB) 2000-01-18 US disclosed