SCHEMBL8106501

SCHEMBL8106501

Cc1ccc(C2(C(=O)OC3CCN(C)CC3)CCC2)cc1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SCN1A P35498 1/20 0.57
SCN2A Q99250 1/20 0.57
SCN3A Q9NY46 1/20 0.57
OPRM1 P35372 6/20 0.55
CHRM3 P20309 3/20 0.49
SLC22A1 O15245 1/20 0.44
SLC6A4 P31645 1/20 0.44
ADRA1A P35348 1/20 0.44
OPRD1 P41143 1/20 0.44
OPRK1 P41145 1/20 0.44
KCNH2 Q12809 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
CYP2D6 P10635 1/20 0.43
CHRM4 P08173 1/20 0.43
CHRM5 P08912 1/20 0.43
CHRM1 P11229 1/20 0.43
ATM Q13315 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8112554 0.87 RAB9A (0.54) OPRM1CHRM3KMT2ACHRM5CHRM1
Hydrochloric Acid SCHEMBL8097354 0.87 CHRM3 (0.62) SCN1ASCN2ASCN3AOPRM1CHRM3
SCHEMBL4734246 0.85 CHRM3 (0.67) SCN1ASCN2ASCN3AOPRM1CHRM3
SCHEMBL4734319 0.84 CHRM3 (0.69) SCN1ASCN2ASCN3AOPRM1CHRM3
SCHEMBL4733406 0.84 CHRM3 (0.69) SCN1ASCN2ASCN3AOPRM1CHRM3
Hydrochloric Acid SCHEMBL1805907 0.84 CHRM3 (0.65) SCN1ASCN2ASCN3AOPRM1CHRM3
SCHEMBL4733989 0.84 CHRM3 (0.69) SCN1ASCN2ASCN3AOPRM1CHRM3
Hydrochloric Acid SCHEMBL8110706 0.81 CHRM3 (0.57) OPRM1CHRM3SLC22A1SLC6A4ADRA1A
SCHEMBL14209817 0.78 CHRM3 (0.64) OPRM1CHRM3SLC22A1SLC6A4ADRA1A
Hydrochloric Acid SCHEMBL8110612 0.78 CHRM3 (0.46) SCN1ASCN2ASCN3AOPRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6124354-A TREATMENT OF URINARY INCONTINENCE OR IRRITABLE BOWEL SYNDROME PHARMACIA & UPJOHN AB (SE) 2000-09-26 US disclosed
EP-0923536-A1 ARYLCYCLOALKANE CARBOXYLIC ESTERS, THEIR USE, PHARMACEUTICAL COMPOSITIONS AND PREPARATION Pharmacia & Upjohn Aktiebolag (SE) 1999-06-23 EP disclosed
WO-1998004517-A1 ARYLCYCLOALKANE CARBOXYLIC ESTERS, THEIR USE, PHARMACEUTICAL COMPOSITIONS AND PREPARATION PHARMACIA & UPJOHN AB (SE) 1998-02-05 WO disclosed