SCHEMBL8107748

SCHEMBL8107748

COc1ccc(CCNC(=O)C(OS(C)(=O)=O)c2ccccc2)cc1OC

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.57
ALDH1A1 P00352 4/20 0.57
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
ADRB2 P07550 1/20 0.54
PLAAT3 P53816 1/20 0.54
PLAAT5 Q96KN8 1/20 0.54
PLAAT2 Q9NWW9 1/20 0.54
PLAAT4 Q9UL19 1/20 0.54
MAPT P10636 1/20 0.54
MAPK1 P28482 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
CA12 O43570 1/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
CA9 Q16790 1/20 0.53
HPGD P15428 1/20 0.53
ALOX12 P18054 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
THRB P10828 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10690654 0.88 KMT2A (0.59) ALDH1A1MEN1KMT2AADRB2PLAAT3
SCHEMBL742343 0.83 KMT2A (0.71) ALDH1A1MEN1KMT2AADRB2PLAAT3
SCHEMBL8098635 0.82 ALDH1A1 (0.62) ALDH1A1MEN1KMT2AADRB2PLAAT3
SCHEMBL6094268 0.82 ALDH1A1 (0.62) ALDH1A1MEN1KMT2AADRB2PLAAT3
SCHEMBL11509318 0.81 ALDH1A1 (0.61) HTTALDH1A1MEN1KMT2AADRB2
SCHEMBL8428854 0.81 ALDH1A1 (0.61) ALDH1A1MEN1KMT2AADRB2PLAAT3
SCHEMBL20418416 0.81 ALDH1A1 (0.61) HTTALDH1A1MEN1KMT2AADRB2
SCHEMBL6376353 0.81 POLB (0.68) ALDH1A1MEN1KMT2AADRB2PLAAT3
SCHEMBL2778736 0.78 ALDH1A1 (0.57) ALDH1A1MEN1KMT2AADRB2PLAAT3
SCHEMBL11888467 0.77 GAA (0.65) ALDH1A1MEN1KMT2AMAPTCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6136819-A COMPOUNDS FOR ANTIINFLAMMATORY AGENTS OR CARDIOVASCULAR DISORDERS BOEHRINGER INGELHEIM GMBH (DE) 2000-10-24 US disclosed
US-5968948-A FOR TREATMENT OF EPILEPSY, STROKE, ALZHEIMER'S DISEASE, BRAIN DISEASES OR AS ANTIINFLAMMATORY OR ANTIPROLIFERATIVE AGENTS BOERHINGER INGELHEIM GMBH (DE) 1999-10-19 US disclosed
US-5661157-A Annelated dihydropyridines and the use thereof for preparing pharmaceutical preparations BOEHRINGER INGELHEIM KG (DE) 1997-08-26 US disclosed