SCHEMBL8108014

SCHEMBL8108014

CC(n1c(=O)c(=O)[nH]c2cc([N+](=O)[O-])c(N3CCOCC3)cc21)P(=O)(O)O

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
MAPT P10636 3/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
AKR1B1 P15121 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8342205 0.96 ALDH1A1 (0.40) ALDH1A1MAPTCYP1A2CYP3A4CYP2D6
SCHEMBL8340372 0.87 HTT (0.39) MAPTLMNAHTT
SCHEMBL8340369 0.86 MAPT (0.41) ALDH1A1MAPTLMNAHTT
SCHEMBL8343007 0.83 HTT (0.39) ALDH1A1MAPTLMNAHTT
SCHEMBL8343002 0.83 MAPT (0.41) ALDH1A1MAPTCYP1A2CYP3A4CYP2D6
SCHEMBL8107840 0.82 GRIA1 (0.50)
SCHEMBL8340567 0.81 GRIN1 (0.39) MAPTCYP1A2CYP3A4LMNA
SCHEMBL8342187 0.81 GRIK1 (0.50)
SCHEMBL8340503 0.79 GRIN1 (0.37) MAPTCYP1A2CYP3A4LMNA
SCHEMBL8344895 0.78 GRIA1 (0.50) ALDH1A1MAPTCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696288-B1 QUINOXALINDIONE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN DRUGS SCHERING AG (DE) 2000-09-20 EP claimed
US-5955461-A Quinoxalinedione derivatives, their production and use in pharmaceutical agents SCHERING AKTIENGESELLSCHAFT (DE) 1999-09-21 US claimed
US-5750525-A Quinoxalinedione derivatives, their production and use in pharmaceutical agents SCHERING AKTIENGESELLSCHAFT (DE) 1998-05-12 US claimed
US-5955461-A Quinoxalinedione derivatives, their production and use in pharmaceutical agents SCHERING AKTIENGESELLSCHAFT (DE) 1999-09-21 US disclosed
US-5750525-A Quinoxalinedione derivatives, their production and use in pharmaceutical agents SCHERING AKTIENGESELLSCHAFT (DE) 1998-05-12 US disclosed