SCHEMBL8340503

SCHEMBL8340503

CC(n1c(=O)c(=O)[nH]c2cc(F)c([N+](=O)[O-])cc21)P(=O)(O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 6/20 0.37
GRIN2D O15399 5/20 0.37
GRIN3B O60391 5/20 0.37
GRIN2A Q12879 5/20 0.37
GRIN2B Q13224 5/20 0.37
GRIN2C Q14957 5/20 0.37
GRIN3A Q8TCU5 5/20 0.37
GRIA1 P42261 2/20 0.37
GRIA2 P42262 2/20 0.37
GRIA3 P42263 2/20 0.37
GRIA4 P48058 2/20 0.37
CA1 P00915 1/20 0.37
MMP2 P08253 1/20 0.37
CA14 Q9ULX7 1/20 0.37
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8340567 0.95 GRIN1 (0.39) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B
SCHEMBL8345260 0.85 GRIK1 (0.34) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B
SCHEMBL8345257 0.84 GRIN2D (0.38) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B
SCHEMBL8342205 0.81 ALDH1A1 (0.40) LMNACYP1A2CYP3A4MAPT
SCHEMBL8342152 0.81 GRIK1 (0.36) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B
SCHEMBL8342149 0.80 GRIK1 (0.38) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B
SCHEMBL8108014 0.79 ALDH1A1 (0.40) LMNACYP1A2CYP3A4MAPT
SCHEMBL8342195 0.79 GRIA1 (0.58) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B
SCHEMBL7357704 0.79 GRIA1 (0.46) GRIN1GRIN2DGRIN3BGRIN2AGRIN2B
SCHEMBL8346030 0.79 GRIK1 (0.59) GRIA1GRIA2GRIA3GRIA4GRIK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5955461-A Quinoxalinedione derivatives, their production and use in pharmaceutical agents SCHERING AKTIENGESELLSCHAFT (DE) 1999-09-21 US disclosed
US-5750525-A Quinoxalinedione derivatives, their production and use in pharmaceutical agents SCHERING AKTIENGESELLSCHAFT (DE) 1998-05-12 US disclosed