SCHEMBL8109358

SCHEMBL8109358

COc1cc(F)ccc1OC(C(N)=O)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.47
SLC6A2 P23975 2/20 0.46
SLC6A4 P31645 2/20 0.46
HRH1 P35367 1/20 0.46
SLC6A3 Q01959 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
PPARG P37231 1/20 0.45
PPARA Q07869 1/20 0.45
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 3/20 0.42
LMNA P02545 2/20 0.42
MEN1 O00255 1/20 0.42
ACHE P22303 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
FFAR1 O14842 1/20 0.41
FFAR4 Q5NUL3 1/20 0.41
F9 P00740 2/20 0.41
F10 P00742 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104478 0.89 KMT2A (0.57) KMT2ASLC6A2SLC6A4SLC6A3CYP3A4
SCHEMBL4536442 0.84 KDM4E (0.48) KMT2ASLC6A2SLC6A4HRH1SLC6A3
SCHEMBL17968476 0.78 PPARG (0.52) SLC6A2SLC6A4SLC6A3PPARGPPARA
SCHEMBL11397979 0.78 KMT2A (0.64) KMT2ASLC6A2SLC6A4SLC6A3CYP3A4
SCHEMBL9423730 0.75 KMT2A (0.47) KMT2ASLC6A2SLC6A4HRH1SLC6A3
SCHEMBL30285514 0.75 SMN1; SMN2 (0.48) KMT2ASLC6A2SLC6A4HRH1SLC6A3
SCHEMBL4533785 0.73 KMT2A (0.53) KMT2ASLC6A2SLC6A4SLC6A3CYP3A4
SCHEMBL21881591 0.73 PPARA (0.74) KMT2ASLC6A2SLC6A4SLC6A3PPARG
SCHEMBL9423717 0.72 FFAR1 (0.48) KMT2ACYP3A4CYP2C19LMNAMEN1
SCHEMBL166380 0.72 NFE2L2 (0.61) CYP3A4CYP2C19KDM4EALDH1A1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008122115-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2008-10-16 WO disclosed