SCHEMBL6973954

SCHEMBL6973954

CC(=O)OC(Cc1ccncc1)c1nc(C(C)C)c(Sc2cccc(F)c2)[nH]1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 5/20 0.32
SLC6A9 P48067 4/20 0.32
ADORA3 P0DMS8 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA2B P29275 1/20 0.31
ADORA1 P30542 1/20 0.31
ROCK2 O75116 3/20 0.31
MAPT P10636 1/20 0.31
MAPK13 O15264 1/20 0.31
MAPK12 P53778 1/20 0.31
MAPK11 Q15759 1/20 0.31
MAPK14 Q16539 1/20 0.31
TYMS P04818 1/20 0.31
CDC7 O00311 1/20 0.31
PRKACA P17612 1/20 0.30
KDM4C Q9H3R0 2/20 0.30
LMNA P02545 2/20 0.30
GRM2 Q14416 1/20 0.30
ALDH1A1 P00352 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6957831 0.92 GSK3B (0.30) MAPK14
SCHEMBL6972343 0.90 IDO1 (0.36) MAPTLMNAGRM2ALDH1A1
SCHEMBL7086009 0.90 SLC6A9 (0.30) ROCK1SLC6A9MAPT
SCHEMBL7081545 0.89 CSNK2A2 (0.34) SLC6A9TYMSLMNAALDH1A1L3MBTL1
SCHEMBL6975056 0.89 ALDH1A1 (0.36) ROCK2ALDH1A1L3MBTL1
SCHEMBL6974498 0.88 SLC6A9 (0.35) SLC6A9TYMSLMNAALDH1A1L3MBTL1
SCHEMBL7084827 0.87 SLC6A9 (0.34) SLC6A9ADORA2AADORA1ALDH1A1
SCHEMBL7084286 0.86 MAPK13 (0.30) MAPK13MAPK12MAPK11MAPK14
SCHEMBL8109549 0.86 MAPK14 (0.34) ROCK1SLC6A9ROCK2MAPK13MAPK12
SCHEMBL7078284 0.85 ROCK1 (0.33) ROCK1SLC6A9ADORA3ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed