SCHEMBL8109743

SCHEMBL8109743

CC(C)(C)OC(=O)N1CCC2(CC1)CCN(C(=O)[C@@H]1CCCC[C@H]1C(=O)NC1(C#N)CC1)C2

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSK P43235 19/20 0.51
CTSB P07858 16/20 0.51
CTSS P25774 15/20 0.51
KCNH2 Q12809 5/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13065393 0.82 KMT2A (0.49) CTSKCTSBCTSSKCNH2CYP3A4
SCHEMBL13551798 0.82 KMT2A (0.49) CTSKCTSBCTSSKCNH2CYP3A4
SCHEMBL2241403 0.80 CTSK (0.51) CTSKCTSBCTSSKCNH2CYP3A4
SCHEMBL2241406 0.80 CTSK (0.51) CTSKCTSBCTSSKCNH2CYP3A4
SCHEMBL14642110 0.80 CTSK (0.51) CTSKCTSBCTSSKCNH2CYP3A4
SCHEMBL13064566 0.79 KMT2A (0.49) CTSKCTSBCTSSKCNH2CYP3A4
SCHEMBL4573152 0.75 CTSB (0.67) CTSKCTSBCTSSKCNH2CYP3A4
SCHEMBL13551875 0.74 CTSS (0.43) CTSKCTSBCTSS
SCHEMBL13553343 0.72 CTSS (0.42) CTSKCTSBCTSS
SCHEMBL13552506 0.72 CTSS (0.42) CTSKCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001128-A1 1,2-CYCL0HEXANE DICARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed