SCHEMBL8109939

SCHEMBL8109939

COc1nc(N2CCN(C(=O)OC(C)(C)C)[C@H](C)C2)ccc1C1CC1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.56
HDAC1 Q13547 1/20 0.47
GPR119 Q8TDV5 2/20 0.45
SUV39H2 Q9H5I1 2/20 0.44
CTSB P07858 1/20 0.42
CTSS P25774 1/20 0.42
CTSK P43235 1/20 0.42
PANK3 Q9H999 5/20 0.41
GRM1 Q13255 2/20 0.40
CHRM4 P08173 1/20 0.39
NR1H2 P55055 2/20 0.38
NR1H3 Q13133 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4573828 1.00 MAP4K4 (0.56) MAP4K4HDAC1GPR119SUV39H2CTSB
SCHEMBL4574046 0.86 MAP4K4 (0.59) MAP4K4HDAC1GPR119SUV39H2CTSB
SCHEMBL8097015 0.86 MAP4K4 (0.59) MAP4K4HDAC1GPR119SUV39H2CTSB
SCHEMBL4573074 0.86 CTSB (0.45) MAP4K4CTSBCTSSCTSKPANK3
SCHEMBL4573301 0.85 MAP4K4 (0.58) MAP4K4HDAC1GPR119SUV39H2CTSB
SCHEMBL8117492 0.85 MAP4K4 (0.58) MAP4K4HDAC1GPR119SUV39H2CTSB
SCHEMBL8108991 0.85 GPR119 (0.51) MAP4K4HDAC1GPR119SUV39H2CHRM4
SCHEMBL4573572 0.85 GPR119 (0.51) MAP4K4HDAC1GPR119SUV39H2CHRM4
SCHEMBL16333441 0.84 MAP4K4 (0.57) MAP4K4HDAC1GPR119SUV39H2CTSB
SCHEMBL4573681 0.84 MAP4K4 (0.51) MAP4K4GPR119SUV39H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed