SCHEMBL8110550

SCHEMBL8110550

C=C1CC(CC#N)(c2ccccc2)C1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.40
HTT P42858 1/20 0.40
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
HSD17B10 Q99714 1/20 0.38
DPP4 P27487 1/20 0.36
AXL P30530 1/20 0.36
MERTK Q12866 1/20 0.36
HSD11B1 P28845 1/20 0.33
CCR1 P32246 1/20 0.33
EGFR P00533 1/20 0.33
SLC6A4 P31645 2/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A3 Q01959 1/20 0.33
OPRD1 P41143 1/20 0.32
OPRM1 P35372 3/20 0.32
OPRL1 P41146 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319137 0.77 TSHR (0.53) TSHRHTTMAOAMAOBTAAR1
SCHEMBL8315393 0.77 TSHR (0.57) TSHRHTTMAOAMAOBTAAR1
SCHEMBL19966073 0.76 MAOA (0.44) TSHRHTTMAOAMAOBTAAR1
SCHEMBL2857720 0.76 TSHR (0.55) TSHRHTTMAOAMAOBTAAR1
SCHEMBL13308190 0.75 MAOA (0.42) MAOAMAOBTAAR1DPP4HSD11B1
SCHEMBL15577243 0.73 TSHR (0.42) TSHRHTTMAOAMAOBTAAR1
SCHEMBL15577188 0.73 ICMT (0.43) TSHRHTTMAOAMAOBTAAR1
SCHEMBL8107080 0.73 MAOA (0.46) TSHRHTTMAOAMAOBTAAR1
SCHEMBL5147525 0.73 OPRM1 (0.55) TSHRHTTMAOAMAOBTAAR1
SCHEMBL8317198 0.73 TSHR (0.39) TSHRHTTMAOAMAOBTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6124354-A TREATMENT OF URINARY INCONTINENCE OR IRRITABLE BOWEL SYNDROME PHARMACIA & UPJOHN AB (SE) 2000-09-26 US disclosed
EP-0923536-A1 ARYLCYCLOALKANE CARBOXYLIC ESTERS, THEIR USE, PHARMACEUTICAL COMPOSITIONS AND PREPARATION Pharmacia & Upjohn Aktiebolag (SE) 1999-06-23 EP disclosed
WO-1998004517-A1 ARYLCYCLOALKANE CARBOXYLIC ESTERS, THEIR USE, PHARMACEUTICAL COMPOSITIONS AND PREPARATION PHARMACIA & UPJOHN AB (SE) 1998-02-05 WO disclosed