SCHEMBL8112704

SCHEMBL8112704

CC(C)(C)OC(=O)N[C@H](CCCN/C(N)=N\[N+](=O)[O-])C(=O)NCc1cc(Br)c(N)c(Br)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 6/20 0.46
CA1 P00915 5/20 0.46
CTSK P43235 6/20 0.37
CTSS P25774 5/20 0.37
CXCR3 P49682 2/20 0.37
PARP1 P09874 1/20 0.36
CTSB P07858 1/20 0.36
NPY1R P25929 1/20 0.36
MMP1 P03956 1/20 0.35
MMP3 P08254 1/20 0.35
MMP9 P14780 1/20 0.35
SIRT5 Q9NXA8 1/20 0.35
F2 P00734 1/20 0.35
AAK1 Q2M2I8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8115106 0.90 CA2 (0.44) CA2CA1CTSKCTSSCXCR3
SCHEMBL8112857 0.85 CA2 (0.52) CA2CA1CTSKCTSSNPY1R
SCHEMBL8120447 0.85 CA2 (0.52) CA2CA1CTSKCTSSCXCR3
SCHEMBL8120925 0.84 CA2 (0.51) CA2CA1CTSKCTSSCXCR3
SCHEMBL8114815 0.84 CA2 (0.53) CA2CA1CTSKCTSSCXCR3
SCHEMBL8126119 0.82 CA2 (0.49) CA2CA1CTSKCTSSCXCR3
SCHEMBL7040745 0.82 CA2 (0.49) CA2CA1CTSKCTSSCXCR3
SCHEMBL5966482 0.82 CTSS (0.51) CA2CA1CTSKCTSSCTSB
SCHEMBL8126994 0.81 NPY1R (0.54) NPY1R
SCHEMBL8112106 0.80 CTSK (0.55) CA2CA1CTSKCTSSCXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0680469-B1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME BOEHRINGER INGELHEIM PHARMA (DE) 2000-04-26 EP disclosed