SCHEMBL8113203

SCHEMBL8113203

ON=C1CCN(Cc2ccc(C(F)(F)F)cc2)CC1.ON=C1CCN(Cc2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.61
ALDH1A1 P00352 2/20 0.61
HIF1A Q16665 4/20 0.50
EPAS1 Q99814 4/20 0.50
OPRL1 P41146 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
CHKA P35790 1/20 0.49
POLB P06746 1/20 0.48
GAA P10253 1/20 0.48
FAAH O00519 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
HRH3 Q9Y5N1 1/20 0.46
TEAD1 P28347 1/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
MAPK1 P28482 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6942215 1.00 KDM4E (0.61) KDM4EALDH1A1HIF1AEPAS1OPRL1
SCHEMBL6943510 0.80 ALDH1A1 (0.56) KDM4EALDH1A1POLBGAASIGMAR1
SCHEMBL4145765 0.79 KDM4E (0.67) KDM4EALDH1A1HIF1AEPAS1OPRL1
SCHEMBL8108271 0.79 KDM4E (0.67) KDM4EALDH1A1HIF1AEPAS1OPRL1
SCHEMBL6947935 0.79 HPGD (0.46) KDM4EALDH1A1HIF1APOLBSIGMAR1
SCHEMBL8107724 0.79 HPGD (0.46) KDM4EALDH1A1HIF1APOLBSIGMAR1
SCHEMBL6949777 0.79 ALDH1A1 (0.56) KDM4EALDH1A1L3MBTL1POLBGAA
SCHEMBL8108849 0.79 ALDH1A1 (0.56) KDM4EALDH1A1L3MBTL1POLBGAA
SCHEMBL7270268 0.78 SIGMAR1 (0.61) KDM4EOPRL1L3MBTL1POLBGAA
SCHEMBL21620787 0.78 ALDH1A1 (0.96) KDM4EALDH1A1HIF1AEPAS1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1056744-A1 6,9-DISUBSTITUTED 2- TRANS-(4- AMINOCYCLOHEXYL) AMINO]PURINES Aventis Pharmaceuticals Inc. (US) 2000-12-06 EP disclosed
WO-1999043675-A1 6,9-DISUBSTITUTED 2-[TRANS-(4- AMINOCYCLOHEXYL) AMINO]PURINES AVENTIS PHARMACEUTICALS INC. (US) 1999-09-02 WO disclosed