SCHEMBL8107724

SCHEMBL8107724

ON=C1CCN(Cc2ccncc2)CC1.ON=C1CCN(Cc2ccncc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.46
LSS P48449 1/20 0.46
KDM4E B2RXH2 4/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C9 P11712 2/20 0.46
HIF1A Q16665 1/20 0.46
DRD2 P14416 1/20 0.44
TSHR P16473 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HSD11B1 P28845 1/20 0.43
CASP1 P29466 1/20 0.42
CASP4 P49662 1/20 0.42
CASP5 P51878 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
POLB P06746 1/20 0.41
CCR2 P41597 1/20 0.41
GBA1 P04062 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6947935 1.00 HPGD (0.46) HPGDLSSKDM4EMEN1KMT2A
SCHEMBL7270268 0.82 SIGMAR1 (0.61) KDM4EMEN1KMT2ATSHRSIGMAR1
SCHEMBL6945532 0.81 CHRNB2 (0.64) KDM4EDRD2ALDH1A1CASP1CASP4
SCHEMBL8099634 0.81 CHRNB2 (0.64) KDM4EDRD2ALDH1A1CASP1CASP4
SCHEMBL6943510 0.81 ALDH1A1 (0.56) LSSKDM4EMEN1KMT2ADRD2
SCHEMBL6949777 0.79 ALDH1A1 (0.56) KDM4EMEN1KMT2AALDH1A1POLB
SCHEMBL8108849 0.79 ALDH1A1 (0.56) KDM4EMEN1KMT2AALDH1A1POLB
SCHEMBL28269086 0.79 LSS (0.66) HPGDLSSKDM4EMEN1KMT2A
SCHEMBL8113203 0.79 KDM4E (0.61) KDM4EHIF1AALDH1A1SIGMAR1POLB
SCHEMBL6942215 0.79 KDM4E (0.61) KDM4EHIF1AALDH1A1SIGMAR1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1056744-A1 6,9-DISUBSTITUTED 2- TRANS-(4- AMINOCYCLOHEXYL) AMINO]PURINES Aventis Pharmaceuticals Inc. (US) 2000-12-06 EP disclosed
WO-1999043675-A1 6,9-DISUBSTITUTED 2-[TRANS-(4- AMINOCYCLOHEXYL) AMINO]PURINES AVENTIS PHARMACEUTICALS INC. (US) 1999-09-02 WO disclosed