SCHEMBL8115353

SCHEMBL8115353

CCOC(=O)c1ccc(-c2nc[nH]n2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.53
CA1 P00915 2/20 0.53
CA2 P00918 2/20 0.53
CA7 P43166 2/20 0.53
CA9 Q16790 2/20 0.53
CA14 Q9ULX7 2/20 0.53
ESR1 P03372 1/20 0.53
ESR2 Q92731 1/20 0.53
KDM4E B2RXH2 6/20 0.52
RAB9A P51151 5/20 0.52
NPC1 O15118 4/20 0.52
MAPT P10636 3/20 0.52
HSP90AA1 P07900 1/20 0.52
CYP1A2 P05177 2/20 0.51
LMNA P02545 1/20 0.51
CYP3A4 P08684 1/20 0.51
MAOA P21397 1/20 0.51
HPGD P15428 4/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
ALDH1A1 P00352 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4554490 0.82 ALDH1A1 (0.55) CA12CA1CA2CA7CA9
SCHEMBL4635046 0.80 CA12 (0.63) CA12CA1CA2CA7CA9
SCHEMBL16351874 0.79 CA1 (0.73) CA12CA1CA2CA7CA9
SCHEMBL1965326 0.79 CA1 (0.73) CA12CA1CA2CA7CA9
SCHEMBL27771735 0.79 CA12 (0.58) CA12CA1CA2CA7CA9
SCHEMBL87450 0.77 CA1 (0.83) CA12CA1CA2CA7CA9
SCHEMBL22530121 0.77 XDH (0.60) CA12CA1CA2CA7CA9
SCHEMBL3767499 0.76 KDM4E (0.54) KDM4ERAB9ANPC1MAPTHPGD
SCHEMBL4224606 0.76 KDM4E (0.47) KDM4ERAB9ANPC1ALDH1A1PDGFRB
SCHEMBL754148 0.76 KDM4E (0.47) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986551-A1 SULFONAMIDE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Pharmaceutical Company Limited (JP) 2000-03-22 EP disclosed
WO-1998054164-A1 SULFONAMIDE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-12-03 WO disclosed