SCHEMBL8116286

SCHEMBL8116286

Cc1oc(-c2ccccc2)nc1C(O)COc1ccc(CC2SC(=O)NC2=O)nc1

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PPARG P37231 17/20 0.45
PPARA Q07869 9/20 0.45
CYP3A4 P08684 1/20 0.40
RXRA P19793 1/20 0.40
FFAR1 O14842 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL131888 0.89 PPARG (0.55) PPARGPPARACYP3A4FFAR1
SCHEMBL9878823 0.85 PPARG (0.42) PPARGPPARACYP3A4RXRAFFAR1
SCHEMBL8116894 0.82 PPARG (0.48) PPARGPPARACYP3A4RXRAFFAR1
SCHEMBL10366694 0.81 MAOB (0.47) PPARGPPARACYP3A4FFAR1
SCHEMBL8323757 0.81 PPARG (0.46) PPARGPPARACYP3A4RXRAFFAR1
SCHEMBL2572355 0.79 PPARG (0.58) PPARGPPARACYP3A4RXRAFFAR1
SCHEMBL9520977 0.78 PPARG (0.45) PPARGPPARA
SCHEMBL8163904 0.78 PPARG (0.39) PPARGPPARACYP3A4
SCHEMBL10365707 0.76 PPARG (0.61) PPARGPPARACYP3A4RXRAFFAR1
SCHEMBL9879239 0.76 LIPG (0.38) PPARGPPARAFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0751944-B1 THIAZOLIDINES AND OXAZOLIDINES SUBSTITUTED BY A PYRIDINE RING AND THEIR USE AS HYPOGLYCEMIC AGENTS NISSAN CHEMICAL IND LTD (JP) 2000-12-20 EP disclosed
US-5955481-A Pyridine type thiazolidines NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1999-09-21 US disclosed
WO-1995026347-A1 THIAZOLIDINES AND OXAZOLIDINES SUBSTITUTED BY A PYRIDINE RING AND THEIR USE AS HYPOGLYCEMIC AGENTS NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1995-10-05 WO disclosed