SCHEMBL8118693

SCHEMBL8118693

CC(C)(C)[Si](OCC(I)CCC(=O)O)(c1ccccc1)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP1A2 P05177 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
CPA3 P15088 1/20 0.34
CYP3A4 P08684 2/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
FOLH1 Q04609 2/20 0.33
SMYD2 Q9NRG4 2/20 0.32
GAA P10253 1/20 0.32
ADAMTS4 O75173 1/20 0.32
ADAMTS5 Q9UNA0 1/20 0.32
AAK1 Q2M2I8 1/20 0.32
KDM4E B2RXH2 1/20 0.31
TP53 P04637 1/20 0.31
GLA P06280 1/20 0.31
POLB P06746 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9115853 1.00 ALDH1A1 (0.34) ALDH1A1CYP2D6CYP1A2TSHRCYP2C19
SCHEMBL8118695 1.00 ALDH1A1 (0.34) ALDH1A1CYP2D6CYP1A2TSHRCYP2C19
SCHEMBL5026303 0.85 CYSLTR2 (0.37) ALDH1A1CYP2D6CYP1A2TSHRCYP2C19
SCHEMBL5026306 0.85 CYSLTR2 (0.37) ALDH1A1CYP2D6CYP1A2TSHRCYP2C19
SCHEMBL9523633 0.85 GAA (0.36) ALDH1A1CYP2D6CYP1A2TSHRCYP2C19
SCHEMBL8122701 0.85 GAA (0.36) ALDH1A1CYP2D6CYP1A2TSHRCYP2C19
SCHEMBL8122702 0.85 GAA (0.36) ALDH1A1CYP2D6CYP1A2TSHRCYP2C19
SCHEMBL3404476 0.84 LTA4H (0.38) ALDH1A1CYP2D6CYP1A2TSHRCYP2C19
SCHEMBL9123979 0.80 SMYD2 (0.32) ALDH1A1CYP2D6CYP1A2TSHRCYP2C19
SCHEMBL8116571 0.80 SMYD2 (0.32) ALDH1A1CYP2D6CYP1A2TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0707481-B1 L-2',3'-DIDEOXY NUCLEOSIDE ANALOGS AS ANTI-HEPATITIS B (HBV) AND ANTI-HIV AGENTS UNIV YALE (US) 2000-08-16 EP disclosed
US-5830881-A L-2'3',dideoxy nucleoside analogs as anti-hepatitus B (HBV) agents YALE UNIVERSITY (US) 1998-11-03 US disclosed
US-5631239-A VIRICIDES FOR HEPATITIS YALE UNIVERSITY (US) 1997-05-20 US disclosed
US-5627160-A L-2',3'-dideoxy nucleoside analogs as anti-hepatitis B (HBV) and anti-HIV agents YALE UNIVERSITY (US) 1997-05-06 US disclosed
US-5561120-A LOW TOXICITY TO HOST CELLS YALE UNIVERSITY (US) 1996-10-01 US disclosed
EP-0707481-A4 1996-05-29 EP disclosed
EP-0707481-A1 L-2',3'-DIDEOXY NUCLEOSIDE ANALOGS AS ANTI-HEPATITIS B (HBV) AND ANTI-HIV AGENTS YALE UNIVERSITY (US) 1996-04-24 EP disclosed
WO-1994027616-A1 L-2',3'-DIDEOXY NUCLEOSIDE ANALOGS AS ANTI-HEPATITIS B (HBV) AND ANTI-HIV AGENTS YALE UNIVERSITY (US) 1994-12-08 WO disclosed