SCHEMBL8123261

SCHEMBL8123261

CCOC(=O)CCCC[C@@]1(C(=O)OC(C)(C)C)CCCN1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ARG1 P05089 1/20 0.39
ARG2 P78540 1/20 0.39
CYP1A2 P05177 2/20 0.35
TSHR P16473 2/20 0.34
ALDH1A1 P00352 2/20 0.34
ALOX15 P16050 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
CYP3A4 P08684 1/20 0.34
HSD17B10 Q99714 1/20 0.34
NR1I2 O75469 1/20 0.33
PGR P06401 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
PTGS2 P35354 1/20 0.33
PDE4D Q08499 1/20 0.33
GAA P10253 1/20 0.32
EPHX2 P34913 2/20 0.32
USP2 O75604 1/20 0.32
KMT2A Q03164 2/20 0.32
CYP2D6 P10635 2/20 0.31
SLC6A2 P23975 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8106291 0.91 CYP2D6 (0.33) ARG1ARG2CYP1A2TSHRALDH1A1
SCHEMBL8123993 0.80 ARG1 (0.42) ARG1ARG2CYP2D6SLC6A2SLC6A4
SCHEMBL8116636 0.79 ARG1 (0.40) ARG1ARG2CYP2D6SLC6A2SLC6A4
SCHEMBL16757166 0.78 MGAM (0.36) ARG1ARG2CYP1A2TSHRALOX15
SCHEMBL6170436 0.72 ARG1 (0.37) ARG1ARG2CYP2D6SLC6A2SLC6A4
SCHEMBL17395338 0.72 ARG1 (0.37) ARG1ARG2CYP2D6SLC6A2SLC6A4
SCHEMBL8115611 0.71 CA12 (0.41) ARG1ARG2TDP1
SCHEMBL17393299 0.71 SLC6A4 (0.47) ARG1ARG2ALDH1A1ALOX15TDP1
SCHEMBL27643221 0.70 CYP1A2 (0.55) CYP1A2TSHRALDH1A1ALOX15TDP1
Hydrochloric Acid SCHEMBL17393298 0.70 CYP2D6 (0.46) ARG1ARG2ALOX15KMT2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1056733-A1 HISTAMINE H3 RECEPTOR LIGANDS JAMES BLACK FOUNDATION LIMITED (GB) 2000-12-06 EP disclosed
WO-1999042458-A1 HISTAMINE H3 RECEPTOR LIGANDS JAMES BLACK FOUNDATION LIMITED (GB) 1999-08-26 WO disclosed