SCHEMBL8123733

SCHEMBL8123733

Cc1cc(N=C(N)S)ccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UHRF1 Q96T88 1/20 0.42
PLAU P00749 4/20 0.41
ADRA2A P08913 2/20 0.38
ADRA2B P18089 2/20 0.38
ADRA2C P18825 2/20 0.38
CCNC P24863 2/20 0.36
CDK8 P49336 2/20 0.36
PIK3CB P42338 1/20 0.36
NOS1 P29475 2/20 0.35
PLG P00747 1/20 0.35
HTR3E A5X5Y0 3/20 0.35
HTR3B O95264 3/20 0.35
HTR3A P46098 3/20 0.35
HTR3D Q70Z44 3/20 0.35
HTR3C Q8WXA8 3/20 0.35
MAP4K4 O95819 1/20 0.34
DYRK1A Q13627 1/20 0.33
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4021873 0.78 TRPA1 (0.49) PLAUADRA2AADRA2BADRA2CCCNC
SCHEMBL6953872 0.74 SMN1; SMN2 (0.38) UHRF1SMARCA2SMARCA4
SCHEMBL6953869 0.74 SMN1; SMN2 (0.38) UHRF1SMARCA2SMARCA4
SCHEMBL1703486 0.71 PLG (0.67) PLAUNOS1PLGHTR3EHTR3B
SCHEMBL10666080 0.71
SCHEMBL20194903 0.70
SCHEMBL15881207 0.65 UHRF1 (0.45) UHRF1DYRK1A
SCHEMBL15426999 0.65 UHRF1 (0.45) UHRF1DYRK1A
SCHEMBL16462334 0.65 CYP3A4 (0.48) UHRF1CCNCCDK8PIK3CBDYRK1A
SCHEMBL4003603 0.64 UHRF1 (0.43) UHRF1PLAUCCNCCDK8PIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0984936-A1 CYANOGUANIDINES AS CELL PROLIFERATION INHIBITORS LEO PHARMACEUTICAL PRODUCTS LTD. A/S (LOVENS KEMISKE FABRIK PRODUKTIONSAKTIESELSKAB) (DK) 2000-03-15 EP disclosed
WO-1998054141-A1 CYANOGUANIDINES AS CELL PROLIFERATION INHIBITORS Leo Pharmaceutical Products Ltd. A/S (Løvens Kemiske Fabrik Produktionsaktieselskab) (DK) 1998-12-03 WO disclosed