SCHEMBL8125309

SCHEMBL8125309

Bc1cnc(N)c(S(=O)(=O)Nc2ccc(O)c(O)c2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
PKLR P30613 1/20 0.49
SHMT2 P34897 1/20 0.46
NPC1 O15118 1/20 0.43
PLA2G1B P04054 1/20 0.41
ATG4B Q9Y4P1 1/20 0.41
PIK3C3 Q8NEB9 1/20 0.40
PIK3CD O00329 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
PIK3CG P48736 1/20 0.39
ALDH1A1 P00352 5/20 0.38
HSD17B10 Q99714 2/20 0.37
ALPL P05186 1/20 0.37
GAA P10253 1/20 0.36
GFER P55789 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
HPGD P15428 1/20 0.36
PFKFB3 Q16875 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14023926 0.84 MEN1 (0.69) MEN1KMT2APKLRSHMT2NPC1
SCHEMBL14023880 0.70 FEN1 (0.42) MEN1KMT2APIK3C3PIK3CDPIK3CA
SCHEMBL10079156 0.67 SERPINE1 (0.66) MEN1KMT2APKLRALDH1A1GAA
SCHEMBL8114928 0.67 NPC1 (0.33) MEN1KMT2ANPC1PLA2G1BATG4B
SCHEMBL8127591 0.66 SMN1; SMN2 (0.50) NPC1PIK3C3ALDH1A1HTT
SCHEMBL9953246 0.64 NPC1 (0.68) MEN1KMT2ASHMT2NPC1PLA2G1B
SCHEMBL17792911 0.63 SHMT2 (1.00) MEN1KMT2ASHMT2NPC1PLA2G1B
SCHEMBL13265977 0.63 PKLR (0.46) MEN1KMT2APKLRALDH1A1PFKFB3
SCHEMBL6087365 0.63 CA1 (0.58) PKLRGAAGFERAPOBEC3GHTT
SCHEMBL742688 0.63 NPC1 (0.67) MEN1KMT2ASHMT2NPC1PLA2G1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008144463-A1 QUINOLINE DERIVATIVES AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-11-27 WO disclosed