SCHEMBL8129271

SCHEMBL8129271

Cn1cc(CC2CCN(Cc3ccccc3)C2)c2cc(C#N)ccc21

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.47
BCHE P06276 2/20 0.47
THRB P10828 1/20 0.44
HRH3 Q9Y5N1 1/20 0.43
SLC6A4 P31645 7/20 0.42
HTR1A P08908 3/20 0.42
DRD2 P14416 1/20 0.42
DRD3 P35462 1/20 0.42
CCR3 P51677 2/20 0.42
CHRM2 P08172 2/20 0.42
SLC6A2 P23975 1/20 0.41
SLC6A3 Q01959 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8131620 0.84 ACHE (0.49) ACHEBCHESLC6A4HTR1ADRD2
SCHEMBL8119111 0.83 BCHE (0.48) ACHEBCHECCR3
SCHEMBL8124394 0.79 BCHE (0.51) ACHEBCHEHTR1A
SCHEMBL6214011 0.78 SLC6A4 (0.61) ACHESLC6A4HTR1ADRD2DRD3
SCHEMBL8130052 0.78 ACHE (0.50) ACHEBCHEDRD2
SCHEMBL8119499 0.78 BCHE (0.46) ACHEBCHEHTR1ACCR3
SCHEMBL8124392 0.77 BCHE (0.45) ACHEBCHECCR3
SCHEMBL8129045 0.76 BCHE (0.45) ACHEBCHEDRD2CCR3
SCHEMBL8129042 0.76 BCHE (0.45) ACHEBCHEDRD2CCR3
SCHEMBL8132943 0.76 BCHE (0.49) ACHEBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0610134-B1 Indole derivatives as 5-HT1-like agonists ADIR (FR) 2000-04-05 EP disclosed
US-5348968-A Migraines ADIR ET COMPAGNIE (FR) 1994-09-20 US disclosed
EP-0610134-A1 Indole, indazole and benzisoxazole derivatives as 5-HT1-like agonists ADIR ET COMPAGNIE (FR) 1994-08-10 EP disclosed