SCHEMBL8133013

SCHEMBL8133013

Fc1ccc([N]c2c(Cl)cccc2Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SLC22A2 O15244 1/20 0.35
SLC22A1 O15245 1/20 0.35
SLC22A3 O75751 1/20 0.35
PLAU P00749 1/20 0.35
NOS3 P29474 2/20 0.34
NOS1 P29475 2/20 0.34
MPI P34949 1/20 0.34
TSHR P16473 2/20 0.33
LMNA P02545 2/20 0.33
CYP19A1 P11511 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2A6 P11509 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
ALOX12 P18054 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4083032 0.75 CYP1A2 (0.47) MAPTTSHRLMNACYP1A2CYP2A6
SCHEMBL3181838 0.72 SLC22A2 (0.50) MAPTRAB9ASLC22A2SLC22A1SLC22A3
SCHEMBL5467199 0.69 MIF (0.41) NPC1RAB9ATSHRLMNACYP1A2
SCHEMBL4396878 0.69 NFE2L2 (0.44) MAPTNPC1RAB9ASLC22A2SLC22A1
SCHEMBL20108650 0.65 TYMP (0.42) NPC1RAB9ANOS3TSHRLMNA
SCHEMBL11404060 0.64 NPC1 (0.53) MAPTNPC1RAB9AMEN1KMT2A
SCHEMBL11404058 0.64 NPC1 (0.53) MAPTNPC1RAB9AMEN1KMT2A
SCHEMBL10387393 0.62 MEN1 (0.43) MAPTNPC1RAB9ALMNACYP1A2
SCHEMBL8155665 0.62 TAAR1 (0.41) TSHRLMNACYP1A2CYP2A6MEN1
SCHEMBL10816322 0.62 RAB9A (0.43) MAPTNPC1RAB9ASLC22A2SLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6147080-A PROTEIN KINASE INHIBITORS; ANTIPROLIFERATIVE AGENT VERTEX PHARMACEUTICALS INCORPORATED (US) 2000-11-14 US disclosed