SCHEMBL8133161

SCHEMBL8133161

CCCCCCCN1CCC(CCCc2ccnc3ccc(OCCN)cc23)CC1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR8 P51685 1/20 0.45
KCNH2 Q12809 4/20 0.43
HRH3 Q9Y5N1 7/20 0.40
CYP2D6 P10635 2/20 0.38
HTR1A P08908 5/20 0.38
HTR1D P28221 5/20 0.38
HTR1B P28222 5/20 0.38
KDM4E B2RXH2 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
HTR2A P28223 1/20 0.38
MAPK1 P28482 1/20 0.38
CYP2C19 P33261 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6975728 0.89 CCR8 (0.56) CCR8KCNH2
SCHEMBL6969343 0.87 CCR8 (0.42) CCR8KCNH2CYP2D6HTR1AHTR1D
SCHEMBL6970280 0.84 CCR8 (0.44) CCR8KCNH2CYP2D6HTR1AHTR1D
SCHEMBL6974682 0.83 CCR8 (0.43) CCR8KCNH2HRH3CYP2D6HTR1A
SCHEMBL6972423 0.83 CCR8 (0.43) CCR8KCNH2HRH3CYP2D6HTR1A
SCHEMBL6968017 0.81 CCR8 (0.44) CCR8KCNH2HRH3CYP2D6HTR1A
SCHEMBL6966012 0.79 CCR8 (0.42) CCR8KCNH2CYP2D6HTR1AKDM4E
SCHEMBL6626735 0.78 CCR8 (0.54) CCR8KCNH2HTR1A
SCHEMBL6971729 0.76 CCR8 (0.52) CCR8KCNH2CYP2D6HTR1AKDM4E
SCHEMBL6978601 0.76 CCR8 (0.39) CCR8KCNH2CYP2D6KDM4ECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051413-A1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2000-11-15 EP claimed
WO-1999037635-A1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 1999-07-29 WO claimed