SCHEMBL6978601

SCHEMBL6978601

CCCCCCCN1CC[C@@H](CCCc2ccnc3ccc(OCCCNC(=N)N)cc23)[C@@H](CC)C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR8 P51685 1/20 0.39
MTNR1A P48039 5/20 0.38
MTNR1B P49286 3/20 0.38
SCN1A P35498 1/20 0.37
SCN2A Q99250 1/20 0.37
SCN3A Q9NY46 1/20 0.37
KCNH2 Q12809 4/20 0.35
SLC2A1 P11166 1/20 0.34
CYP2D6 P10635 4/20 0.34
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 3/20 0.34
HPGD P15428 3/20 0.34
HSD17B10 Q99714 3/20 0.34
TSHR P16473 1/20 0.34
MEN1 O00255 1/20 0.34
CYP3A4 P08684 1/20 0.34
KMT2A Q03164 1/20 0.34
CHRM2 P08172 1/20 0.34
ADRA2A P08913 1/20 0.34
SLC6A4 P31645 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6968017 0.89 CCR8 (0.44) CCR8MTNR1AMTNR1BSCN1ASCN2A
SCHEMBL6966012 0.88 CCR8 (0.42) CCR8MTNR1AMTNR1BSCN1ASCN2A
SCHEMBL6969343 0.88 CCR8 (0.42) CCR8MTNR1AMTNR1BSCN1ASCN2A
SCHEMBL6970280 0.88 CCR8 (0.44) CCR8MTNR1AMTNR1BSCN1ASCN2A
SCHEMBL6974682 0.87 CCR8 (0.43) CCR8SCN1ASCN2ASCN3AKCNH2
SCHEMBL6972423 0.87 CCR8 (0.43) CCR8SCN1ASCN2ASCN3AKCNH2
SCHEMBL6971729 0.84 CCR8 (0.52) CCR8MTNR1AMTNR1BKCNH2SLC2A1
SCHEMBL6965739 0.81 DRD3 (0.45) CCR8
SCHEMBL8131415 0.81 SIGMAR1 (0.44) CCR8
SCHEMBL6977691 0.81 CCR8 (0.40) CCR8MTNR1AMTNR1BKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051413-B1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2003-06-04 EP claimed
EP-1051413-A1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2000-11-15 EP disclosed
WO-1999037635-A1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 1999-07-29 WO disclosed