SCHEMBL8136998

SCHEMBL8136998

CS(=O)(=O)Nc1ccc(-c2nnc(N)s2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.56
ALDH1A1 P00352 4/20 0.56
LMNA P02545 3/20 0.56
TP53 P04637 3/20 0.52
KDM4E B2RXH2 9/20 0.51
MGAM O43451 4/20 0.51
GAA P10253 4/20 0.51
SI P14410 4/20 0.51
MGAM2 Q2M2H8 4/20 0.51
NOTUM Q6P988 1/20 0.51
RAB9A P51151 6/20 0.51
NPC1 O15118 4/20 0.51
HPGD P15428 4/20 0.51
HSD17B10 Q99714 3/20 0.51
MAPT P10636 2/20 0.51
CSNK2A2 P19784 1/20 0.50
CSNK2B P67870 1/20 0.50
CSNK2A1 P68400 1/20 0.50
KIF11 P52732 1/20 0.47
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17713894 0.79 ALDH1A1 (0.61) SMN1; SMN2ALDH1A1LMNATP53KDM4E
SCHEMBL19549074 0.78 ALDH1A1 (0.59) SMN1; SMN2ALDH1A1LMNATP53KDM4E
SCHEMBL17725683 0.76 ALDH1A1 (0.57) SMN1; SMN2ALDH1A1LMNATP53KDM4E
SCHEMBL17725684 0.74 ALDH1A1 (0.54) SMN1; SMN2ALDH1A1LMNATP53KDM4E
SCHEMBL11370829 0.73 SMN1; SMN2 (0.57) SMN1; SMN2ALDH1A1LMNATP53KDM4E
SCHEMBL31041151 0.73 KIF11 (0.79) SMN1; SMN2ALDH1A1LMNAKDM4EHPGD
SCHEMBL2497654 0.72 KIF11 (0.66) SMN1; SMN2ALDH1A1LMNAKDM4EHPGD
SCHEMBL6902047 0.72 ALDH1A1 (1.00) SMN1; SMN2ALDH1A1LMNATP53KDM4E
SCHEMBL22181853 0.72 KDM4E (0.57) SMN1; SMN2ALDH1A1LMNATP53KDM4E
SCHEMBL125639 0.72 HPGD (0.73) SMN1; SMN2ALDH1A1LMNATP53KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054876-A1 1,3,4-THIADIAZOLES DERIVATIVES AS KYN-OH INHIBITORS PHARMACIA & UPJOHN S.p.A. (IT) 2000-11-29 EP disclosed
WO-1999028309-A1 1,3,4-THIADIAZOLES DERIVATIVES AS KYN-OH INHIBITORS PHARMACIA & UPJOHN S.P.A. (IT) 1999-06-10 WO disclosed