SCHEMBL8137202

SCHEMBL8137202

O=C(O)C1C=Cc2ccccc2NC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.37
GAA P10253 2/20 0.37
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
ALDH1A1 P00352 2/20 0.34
HSPA1A P0DMV8 1/20 0.33
PTPN7 P35236 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
P2RX4 Q99571 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
EPHX2 P34913 1/20 0.31
HPGD P15428 1/20 0.31
RAB9A P51151 2/20 0.30
NPC1 O15118 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C19 P33261 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
KDM4E B2RXH2 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6632184 0.81 MAPT (0.33) MAPTGAAALDH1A1HSPA1APTPN7
SCHEMBL6628775 0.71 SIRT1 (0.32) MAPTGAAALDH1A1KDM4E
SCHEMBL11498471 0.71
SCHEMBL385982 0.70 MAPT (0.40) MAPTGAAALDH1A1HSPA1APTPN7
SCHEMBL11205813 0.70 GAA (0.40) MAPTGAAALDH1A1P2RX4MEN1
Hydrochloric Acid SCHEMBL7435031 0.69 MAPT (0.39) MAPTGAAALDH1A1HSPA1APTPN7
SCHEMBL5800011 0.68 ALDH1A1 (0.57) MAPTGAAALDH1A1HSPA1APTPN7
SCHEMBL3749720 0.68 ALDH1A1 (0.57) MAPTGAAALDH1A1HSPA1APTPN7
Hydrochloric Acid SCHEMBL28797396 0.67 ALDH1A1 (0.56) MAPTGAAALDH1A1HSPA1APTPN7
Hydrochloric Acid SCHEMBL28270652 0.67 ALDH1A1 (0.56) MAPTGAAALDH1A1HSPA1APTPN7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1649847-A Method for producing optically active sulfoxide derivative TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2005-08-03 CN disclosed
EP-1039899-A2 PHARMACEUTICAL COMPOSITION FOR ANTAGONIZING CCR5 COMPRISING ANILIDE DERIVATIVE Takeda Chemical Industries, Ltd. (JP) 2000-10-04 EP disclosed
WO-1999032100-A2 PHARMACEUTICAL COMPOSITION FOR ANTAGONIZING CCR5 COMPRISING ANILIDE DERIVATIVE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-07-01 WO disclosed